SCHEMBL5260503

SCHEMBL5260503

Cc1c(C(=O)Nc2ccc(Cl)cc2)sc(NC(=O)C(F)(F)F)c1C(C)C

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ANO1 Q5XXA6 7/20 0.50
SMN1; SMN2 Q16637 4/20 0.44
MAPT P10636 4/20 0.44
TP53 P04637 2/20 0.44
MEN1 O00255 2/20 0.44
HPGD P15428 2/20 0.44
KMT2A Q03164 2/20 0.44
AHR P35869 1/20 0.42
F10 P00742 2/20 0.41
PDK1 Q15118 1/20 0.41
PDK2 Q15119 1/20 0.41
PDK3 Q15120 1/20 0.41
PDK4 Q16654 1/20 0.41
NPC1 O15118 1/20 0.40
LMNA P02545 1/20 0.40
RAB9A P51151 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4150011 0.84 MEN1 (0.52) ANO1SMN1; SMN2MAPTTP53MEN1
SCHEMBL4147196 0.74 ANO1 (0.53) ANO1SMN1; SMN2MAPTTP53MEN1
SCHEMBL5550330 0.72 HDAC1 (0.67) ANO1MAPTTP53MEN1KMT2A
SCHEMBL4135317 0.70 ANO1 (0.53) ANO1SMN1; SMN2MAPTMEN1KMT2A
SCHEMBL14366827 0.70 HPGD (0.67) SMN1; SMN2MAPTTP53MEN1HPGD
SCHEMBL11097805 0.68 KIF11 (0.54) SMN1; SMN2MAPTMEN1HPGDKMT2A
SCHEMBL4147246 0.67 ANO1 (0.98) ANO1SMN1; SMN2MAPTTP53
SCHEMBL4134799 0.67 ANO1 (1.00) ANO1SMN1; SMN2MAPTTP53
SCHEMBL4151223 0.67 ANO1 (1.00) ANO1SMN1; SMN2MAPTTP53
SCHEMBL4147414 0.65 ANO1 (0.66) ANO1SMN1; SMN2MAPTTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1802634-A2 THIOPHENS AND THEIR USE AS ANTI-TUMOR AGENTS Compass Pharmaceuticals LLC (US) 2007-07-04 EP claimed
WO-2006044826-A2 THIOPHENS AND THEIR USE AS ANTI-TUMOR AGENTS COMPASS PHARMACEUTICALS LLC (US) 2006-04-27 WO claimed
EP-1802634-A2 THIOPHENS AND THEIR USE AS ANTI-TUMOR AGENTS Compass Pharmaceuticals LLC (US) 2007-07-04 EP disclosed
WO-2006044826-A2 THIOPHENS AND THEIR USE AS ANTI-TUMOR AGENTS COMPASS PHARMACEUTICALS LLC (US) 2006-04-27 WO disclosed