SCHEMBL5260591

SCHEMBL5260591

CC(NC(=O)c1ccc(-c2nnn[nH]2)cc1)C(Cc1ccc(Cl)cc1)c1ccc(Cl)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 16/20 0.48
CNR2 P34972 12/20 0.48
FDFT1 P37268 2/20 0.47
ROCK2 O75116 1/20 0.43
PRKACA P17612 1/20 0.43
RPS6KB1 P23443 1/20 0.43
IRAK1 P51617 1/20 0.43
PRKX P51817 1/20 0.43
LIMK1 P53667 1/20 0.43
PRKG2 Q13237 1/20 0.43
ROCK1 Q13464 1/20 0.43
PRKG1 Q13976 1/20 0.43
PKN2 Q16513 1/20 0.43
HIPK4 Q8NE63 1/20 0.43
AURKB Q96GD4 1/20 0.43
CLK4 Q9HAZ1 1/20 0.43
CSNK1G1 Q9HCP0 1/20 0.43
MEN1 O00255 1/20 0.42
RAB9A P51151 1/20 0.42
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5260356 0.88 CNR1 (0.52) CNR1CNR2FDFT1
SCHEMBL5262269 0.83 CNR1 (0.63) CNR1CNR2FDFT1MEN1RAB9A
SCHEMBL5262358 0.83 CNR1 (0.46) CNR1CNR2FDFT1
SCHEMBL5260602 0.81 CNR1 (0.44) CNR1CNR2FDFT1
SCHEMBL5260009 0.80 FDFT1 (0.68) CNR1CNR2FDFT1
SCHEMBL5260594 0.79 RAB9A (0.44) MEN1RAB9AKMT2ASMN1; SMN2
SCHEMBL5265148 0.78 CNR1 (0.53) CNR1CNR2FDFT1
SCHEMBL5262390 0.78 CNR1 (0.59) CNR1CNR2FDFT1ROCK2PRKACA
SCHEMBL5262773 0.78 CNR1 (0.72) CNR1CNR2FDFT1
SCHEMBL5261389 0.75 CNR1 (0.55) CNR1CNR2FDFT1ROCK2PRKACA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1494997-A4 SUBSTITUTED ARYL AMIDES MERCK & CO INC (US) 2007-04-11 EP claimed
JP-2005527586-A 2005-09-15 JP claimed
EP-1494997-A1 SUBSTITUTED ARYL AMIDES Merck & Co., Inc. (US) 2005-01-12 EP claimed
WO-2003087037-A1 SUBSTITUTED ARYL AMIDES MERCK & CO., INC. (US) 2003-10-23 WO claimed
EP-1494997-A4 SUBSTITUTED ARYL AMIDES MERCK & CO INC (US) 2007-04-11 EP disclosed
EP-1494997-A1 SUBSTITUTED ARYL AMIDES Merck & Co., Inc. (US) 2005-01-12 EP disclosed
WO-2003087037-A1 SUBSTITUTED ARYL AMIDES MERCK & CO., INC. (US) 2003-10-23 WO disclosed