SCHEMBL5260640

SCHEMBL5260640

CC(CNCC(COc1ccc(-c2nc3cc(Br)cnc3[nH]2)cc1)OC(=O)C(F)(F)F)OC(=O)C(F)(F)F

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 1/20 0.34
MMP2 P08253 1/20 0.33
MMP9 P14780 1/20 0.33
MMP8 P22894 1/20 0.33
MMP13 P45452 1/20 0.33
HDAC6 Q9UBN7 5/20 0.33
HDAC3 O15379 4/20 0.33
HDAC1 Q13547 4/20 0.33
HDAC2 Q92769 4/20 0.33
HDAC8 Q9BY41 4/20 0.33
HDAC4 P56524 3/20 0.33
HDAC7 Q8WUI4 3/20 0.33
HDAC10 Q969S8 3/20 0.33
HDAC11 Q96DB2 3/20 0.33
HDAC9 Q9UKV0 3/20 0.33
HDAC5 Q9UQL6 3/20 0.33
TRPV1 Q8NER1 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4838292 0.87 HDAC3 (0.34) CHEK2MMP2MMP9MMP8MMP13
SCHEMBL4834997 0.86 HDAC6 (0.36) CHEK2HDAC6HDAC3HDAC1HDAC2
SCHEMBL4843544 0.86 CHEK2 (0.34) CHEK2MMP2MMP9MMP8MMP13
SCHEMBL4840576 0.81 HDAC6 (0.35) CHEK2HDAC6HDAC3HDAC1HDAC2
Trifluoroacetic Acid SCHEMBL5260635 0.80
SCHEMBL4841843 0.79 CHEK2 (0.32) CHEK2HDAC6HDAC3HDAC1HDAC2
SCHEMBL4845811 0.78 NPC1 (0.35) CHEK2HDAC6
SCHEMBL4844169 0.78 CHEK2 (0.37) CHEK2
SCHEMBL4839425 0.78 CHEK2 (0.35) CHEK2HDAC6
SCHEMBL4842378 0.77 CHEK2 (0.38) CHEK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539759-B1 NOVEL IMIDAZOPYRIDINES AND THEIR USE ASTRAZENECA AB (SE) 2007-08-15 EP disclosed