SCHEMBL526216

SCHEMBL526216

C=CCc1ccc(OC(CCNC)c2ccccc2)c(-c2cc(CC=C)ccc2OC(F)(F)F)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 11/20 0.48
SLC6A2 P23975 9/20 0.46
CYP2D6 P10635 8/20 0.46
CYP3A4 P08684 6/20 0.46
KMT2A Q03164 6/20 0.46
CYP1A2 P05177 5/20 0.46
SLC6A3 Q01959 5/20 0.46
MEN1 O00255 5/20 0.46
LMNA P02545 5/20 0.46
PMP22 Q01453 5/20 0.46
TSHR P16473 4/20 0.46
HTR2C P28335 4/20 0.46
CHRM1 P11229 3/20 0.46
ADRA2B P18089 3/20 0.46
HTR2A P28223 3/20 0.46
HRH1 P35367 3/20 0.46
OPRM1 P35372 3/20 0.46
OPRK1 P41145 3/20 0.46
HTR2B P41595 3/20 0.46
KCNH2 Q12809 3/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL525549 0.88 SLC6A4 (0.59) SLC6A4SLC6A2CYP2D6CYP3A4KMT2A
Hydrochloric Acid SCHEMBL725835 0.87 SLC6A2 (0.60) SLC6A4SLC6A2CYP2D6CYP3A4KMT2A
SCHEMBL525534 0.86 GABRA1 (0.54) SLC6A4SLC6A2CYP2D6CYP3A4KMT2A
SCHEMBL525899 0.86 SLC6A4 (0.52) SLC6A4SLC6A2CYP2D6CYP3A4KMT2A
Hydrochloric Acid SCHEMBL726060 0.85 SLC6A4 (0.51) SLC6A4SLC6A2CYP2D6CYP3A4KMT2A
Hydrochloric Acid SCHEMBL530274 0.85 GABRA1 (0.53) SLC6A4SLC6A2CYP2D6CYP3A4KMT2A
SCHEMBL525738 0.81 SLC6A4 (0.46) SLC6A4SLC6A2CYP2D6CYP3A4KMT2A
Hydrochloric Acid SCHEMBL726038 0.81 NOS2 (0.42) SLC6A4SLC6A2CYP2D6CYP3A4KMT2A
SCHEMBL526594 0.80 NOS2 (0.47) SLC6A4SLC6A2CYP2D6CYP3A4KMT2A
SCHEMBL526595 0.80 NOS2 (0.47) SLC6A4SLC6A2CYP2D6CYP3A4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2423181-A1 Multitarget substituted biphenyl diol derivatives PROUS INSTITUTE FOR BIOMEDICAL RESEARCH S.A. (ES) 2012-02-29 EP claimed
WO-2012013691-A1 MULTITARGET SUBSTITUTED BIPHENYL DIOL DERIVATIVES PROUS INSTITUTE FOR BIOMEDICAL RESEARCH, S.A. (ES) 2012-02-02 WO claimed
EP-2423181-A1 Multitarget substituted biphenyl diol derivatives PROUS INSTITUTE FOR BIOMEDICAL RESEARCH S.A. (ES) 2012-02-29 EP disclosed
WO-2012013691-A1 MULTITARGET SUBSTITUTED BIPHENYL DIOL DERIVATIVES PROUS INSTITUTE FOR BIOMEDICAL RESEARCH, S.A. (ES) 2012-02-02 WO disclosed