SCHEMBL526321

SCHEMBL526321

Oc1ccc(Nc2nc(-c3ccc(Cl)cc3)cs2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 13/20 1.00
VCP P55072 7/20 1.00
AMY1A P0DUB6 4/20 1.00
MAPT P10636 3/20 1.00
ALOX15 P16050 2/20 1.00
TSHR P16473 2/20 1.00
TDP1 Q9NUW8 2/20 1.00
MEN1 O00255 2/20 1.00
MAPK1 P28482 2/20 1.00
KMT2A Q03164 2/20 1.00
DEGS1 O15121 1/20 1.00
MAP4K4 O95819 1/20 1.00
CYP3A4 P08684 1/20 1.00
MAPKAPK2 P49137 1/20 1.00
PIM3 Q86V86 1/20 1.00
MINK1 Q8N4C8 1/20 1.00
SPHK2 Q9NRA0 1/20 1.00
SPHK1 Q9NYA1 1/20 1.00
ALDH1A1 P00352 2/20 0.85
GAA P10253 2/20 0.85

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26125550 1.00 ALOX5 (1.00) ALOX5VCPAMY1AMAPTALOX15
SCHEMBL14825241 0.92 MAPT (1.00) ALOX5VCPAMY1AMAPTALOX15
SCHEMBL12297672 0.85 ALOX5 (0.89) ALOX5VCPAMY1AMAPTALOX15
SCHEMBL12297190 0.85 ALOX5 (0.74) ALOX5VCPAMY1AMAPTALOX15
SCHEMBL2755470 0.85 VCP (1.00) ALOX5VCPAMY1AMAPTALOX15
SCHEMBL12298240 0.85 ALOX5 (0.94) ALOX5VCPAMY1AMAPTALOX15
SCHEMBL1887335 0.85 ESR1 (1.00) ALOX5VCPAMY1AMAPTALOX15
SCHEMBL1822974 0.85 ALOX5 (0.88) ALOX5VCPAMY1AMAPTALOX15
SCHEMBL1882991 0.85 VCP (1.00) ALOX5VCPAMY1AMAPTALOX15
SCHEMBL29152948 0.85 ALOX5 (1.00) ALOX5VCPAMY1AMAPTALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 124 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119300037-A Cross-domain authentication method and system under vehicle-mounted ad hoc network 西安邮电大学 2025-01-10 CN claimed
EP-4181906-A1 SPHINGOID COMPOUNDS FOR USE IN PROPHYLAXIS AND/OR THERAPY OF CORONAVIRIDAE INFECTION Harbins Ruhr Bioscience, Inc. (US) 2023-05-24 EP claimed
US-20230107927-A1 METHODS OF TREATING IATROGENIC AUTOIMMUNE COLITIS FIRST WAVE BIO, INC. 2023-04-06 US claimed
WO-2022015348-A1 SPHINGOID COMPOUNDS FOR USE IN PROPHYLAXIS AND/OR THERAPY OF CORONAVIRIDAE INFECTION Harbins Ruhr Bioscience, Inc. (US) 2022-01-20 WO claimed
EP-3863616-A2 SPHINGOID COMPOUNDS FOR USE IN THE PROPHYLAXIS AND/OR THERAPY OF A VIRAL INFECTION Harbins Ruhr Bioscience, Inc. (US) 2021-08-18 EP claimed
US-20180110757-A1 METHODS OF TREATING PRURITIS AND PAIN THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2018-04-26 US claimed
US-20170252311-A1 SPHINGOSINE KINASE INHIBITORS AND CERAMIDE FOR MAINTENANCE THERAPY OF GLIOBLASTOMA SIGNPATH PHARMA INC. 2017-09-07 US claimed
US-9687477-B2 Modulation of sphingosine 1-phosphate metabolizing enzymes for the treatment of negative-strand RNA virus infections THE CURATORS OF THE UNIVERSITY OF MISSOURI (US) 2017-06-27 US claimed
US-20150126564-A1 MODULATION OF SPHINGOSINE 1-PHOSPHATE METABOLIZING ENZYMES FOR THE TREATMENT OF NEGATIVE-STRAND RNA VIRUS INFECTIONS THE CURATORS OF THE UNIVERSITY OF MISSOURI (US) 2015-05-07 US claimed
US-20140056917-A1 FTY720 Increases CD74 Expression and Sensitizes Cancer Cells to Anti-CD74 Antibody-Mediated Cell Death IMMUNOMEDICS, INC. (US) 2014-02-27 US claimed
WO-2012166859-A2 MODULATION OF SPHINGOSINE 1-PHOSPHATE METABOLIZING ENZYMES FOR THE TREATMENT OF NEGATIVE-STRAND RNA VIRUS INFECTIONS THE CURATORS OF THE UNIVERSITY OF MISSOURI (US) 2012-12-06 WO claimed
US-20120122870-A1 Treatment Of Ischemia-Reperfusion Injury MUSC FOUNDATION FOR RESEARCH DEVELOPMENT (US) 2012-05-17 US claimed
WO-2010129954-A1 TREATMENT OF ISCHEMIA-REPERFUSION INJURY APOGEE BIOTECHNOLOGY CORPORATION (US) 2010-11-11 WO claimed
US-7220764-B2 Such as 5-(2,4-dihydroxy-benzylidene)-3-(4-methoxy-phenyl)-2-thioxo-thiazolidin-4 -one; for treating/preventing hyperproliferative disease, autoimmune disease, inflammatory disease, or allergy THE PENNSYLVANIA STATE UNIVERSITY RESEARCH FOUNDATION (US) 2007-05-22 US claimed
US-20040034075-A1 Sphingosine kinase inhibitors THE PENNSYLVANIA STATE UNIVERSITY RESEARCH FOUNDATION (US) 2004-02-19 US claimed
WO-2003105840-A2 SPHINGOSINE KINASE INHIBITORS THE PENNSYLVANIA STATE RESEARCH FOUNDATION (US) 2003-12-24 WO claimed
WO-2026104911-A1 FAST ANTENNA CALIBRATION BY ORTHOGONAL CARRIER SOUNDING (FACOCS) TEJAS NETWORKS LIMITED (IN) 2026-05-21 WO disclosed
EP-4662319-A2 PERSONALIZED CRISPR PROFILING FOR CANCER Integrate Bioscience LLC (US) 2025-12-17 EP disclosed
US-7220764-B2 Such as 5-(2,4-dihydroxy-benzylidene)-3-(4-methoxy-phenyl)-2-thioxo-thiazolidin-4 -one; for treating/preventing hyperproliferative disease, autoimmune disease, inflammatory disease, or allergy THE PENNSYLVANIA STATE UNIVERSITY RESEARCH FOUNDATION (US) 2007-05-22 US disclosed
WO-2006019586-A2 METHOD OF TREATING TRAUMA OR SEPSIS HAUSER CARL J (US) 2006-02-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120122870-A1 Treatment Of Ischemia-Reperfusion Injury SPHK1, SPHK2, S1PR2 ALOX5 254/4885VCP 3891/4885AMY1A 2663/4885
US-20040034075-A1 Sphingosine kinase inhibitors SPHK1, SPHK2, S1PR1 ALOX5 439/4885VCP 4626/4885AMY1A 3249/4885
US-20180110757-A1 METHODS OF TREATING PRURITIS AND PAIN CYSLTR2, LTB4R2, CYSLTR1 ALOX5 84/4885VCP 3631/4885AMY1A 1956/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.