SCHEMBL526343

SCHEMBL526343

NC(CCO)CNCC(=O)O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRP O00591 2/20 0.40
GABRD O14764 2/20 0.40
GABRA1 P14867 2/20 0.40
GABRB1 P18505 2/20 0.40
GABRG2 P18507 2/20 0.40
GABRB3 P28472 2/20 0.40
GABRA5 P31644 2/20 0.40
GABRA3 P34903 2/20 0.40
GABRA2 P47869 2/20 0.40
GABRB2 P47870 2/20 0.40
GABRA4 P48169 2/20 0.40
GABRE P78334 2/20 0.40
GABRA6 Q16445 2/20 0.40
GABRG1 Q8N1C3 2/20 0.40
GABRG3 Q99928 2/20 0.40
GABRQ Q9UN88 2/20 0.40
ENPEP Q07075 6/20 0.38
ANPEP P15144 3/20 0.38
GRM8 O00222 1/20 0.35
GRM6 O15303 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18583431 0.83 ENPEP (0.35) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL28795088 0.82 ALDH1A1 (0.52) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL8197521 0.80
SCHEMBL31378503 0.79 ALDH1A1 (0.49) ENPEPSLC1A3SLC1A2SLC1A1ALDH1A1
SCHEMBL28648030 0.77 FFAR3 (0.39) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL986003 0.77 PTPN1 (0.40) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL5811235 0.76 ENPEP (0.48) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL1736126 0.76 ALDH1A1 (0.54) ALDH1A1MEN1TSHRKMT2APTPN1
Propionic Acid SCHEMBL18227012 0.76 ALDH1A1 (0.42) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL10924286 0.76

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017189077-A1 HYDROPHILIC SILANES DOW CORNING CORPORATION (US) 2017-11-02 WO disclosed
EP-1895979-B1 COSMETICS COMPRISING A MODIFIED ORGANOPOLYSILOXANE DOW CORNING TORAY CO LTD (JP) 2014-03-12 EP disclosed
EP-2658899-A1 COSMETIC CONTAINING LIQUID ORGANOPOLYSILOXANE Dow Corning Toray Co., Ltd. (JP) 2013-11-06 EP disclosed
EP-2598112-A1 COSMETIC FOR HAIR CONTAINING SUGAR ALCOHOL-MODIFIED SILICONE Dow Corning Toray Co., Ltd. (JP) 2013-06-05 EP disclosed
EP-2598113-A1 COSMETIC FOR HAIR CONTAINING CO-MODIFIED ORGANOPOLYSILOXANE Dow Corning Toray Co., Ltd. (JP) 2013-06-05 EP disclosed
EP-2563327-A1 POWDER TREATMENT AGENT COMPRISING SUGAR ALCOHOL -MODIFIED ORGANOPOLYSILOXANE Dow Corning Toray Co., Ltd. (JP) 2013-03-06 EP disclosed
EP-2563844-A1 ORGANOPOLYSILOXANE AND USE THEREOF AS SURFACTANT, POWDER TREATMENT AGENT, THICKENING AGENT OF OIL -BASED RAW MATERIAL OR GELLING AGENT. GEL AND EMULSION COMPOSITIONS, AS WELL AS, PREPARATIONS FOR EXTERNAL USE AND COSMETICS COMPRISING THE SAME Dow Corning Toray Co., Ltd. (JP) 2013-03-06 EP disclosed
EP-2563845-A1 NOVEL ORGANOPOLYSILOXANE, SURFACTANT, EMULSION COMPOSITION, POWDER TREATMENT AGENT, THICKENING AGENT OF OIL-BASED RAW MATERIAL, GELLING AGENT, GEL COMPOSITION, AND COSMETIC RAW MATERIAL COMPRISING NOVEL ORGANOPOLYSILOXANE, AS WELL AS, PREPARATION FOR EXTERNAL USE AND COSMETIC COMPRISING THE SAME Dow Corning Toray Co., Ltd. (JP) 2013-03-06 EP disclosed
EP-2515841-A1 COPOLYMER HAVING CARBOSILOXANE DENDRIMER STRUCTURE, AND COMPOSITION AND COSMETIC CONTAINING THE SAME Dow Corning Toray Co., Ltd. (JP) 2012-10-31 EP disclosed
EP-2507248-A1 LINEAR AND CYCLIC SILOXANES AND COSMETIC COMPOSITIONS MADE THEREOF Dow Corning Toray Co., Ltd. (JP) 2012-10-10 EP disclosed
WO-2012091155-A1 COSMETIC CONTAINING LIQUID ORGANOPOLYSILOXANE DOW CORNING TORAY CO., LTD. (JP) 2012-07-05 WO disclosed
WO-2012015070-A1 COSMETIC FOR HAIR CONTAINING CO-MODIFIED ORGANOPOLYSILOXANE DOW CORNING TORAY CO., LTD. (JP) 2012-02-02 WO disclosed
WO-2012015069-A1 COSMETIC FOR HAIR CONTAINING SUGAR ALCOHOL-MODIFIED SILICONE DOW CORNING TORAY CO., LTD. (JP) 2012-02-02 WO disclosed
WO-2011136394-A1 POWDER TREATMENT AGENT COMPRISING SUGAR ALCOHOL -MODIFIED ORGANOPOLYSILOXANE DOW CORNING TORAY CO., LTD. (JP) 2011-11-03 WO disclosed
WO-2011136393-A1 ORGANOPOLYSILOXANE AND USE THEREOF AS SURFACTANT, POWDER TREATMENT AGENT, THICKENING AGENT OF OIL -BASED RAW MATERIAL OR GELLING AGENT. GEL AND EMULSION COMPOSITIONS, AS WELL AS, PREPARATIONS FOR EXTERNAL USE AND COSMETICS COMPRISING THE SAME DOW CORNING TORAY CO., LTD. (JP) 2011-11-03 WO disclosed
WO-2011136397-A1 NOVEL ORGANOPOLYSILOXANE, SURFACTANT, EMULSION COMPOSITION, POWDER TREATMENT AGENT, THICKENING AGENT OF OIL-BASED RAW MATERIAL, GELLING AGENT, GEL COMPOSITION, AND COSMETIC RAW MATERIAL COMPRISING NOVEL ORGANOPOLYSILOXANE, AS WELL AS, PREPARATION FOR EXTERNAL USE AND COSMETIC COMPRISING THE SAME DOW CORNING TORAY CO., LTD. (JP) 2011-11-03 WO disclosed
WO-2011078407-A1 COPOLYMER HAVING CARBOSILOXANE DENDRIMER STRUCTURE, AND COMPOSITION AND COSMETIC CONTAINING THE SAME DOW CORNING TORAY CO., LTD. (JP) 2011-06-30 WO disclosed
WO-2011068250-A1 LINEAR AND CYCLIC SILOXANES AND COSMETIC COMPOSITIONS MADE THEREOF DOW CORNING TORAY CO., LTD. (JP) 2011-06-09 WO disclosed
EP-1895979-A1 COSMETICS COMPRISING A MODIFIED ORGANOPOLYSILOXANE Dow Corning Toray Co., Ltd. (JP) 2008-03-12 EP disclosed
WO-2006137576-A1 COSMETICS COMPRISING A MODIFIED ORGANOPOLYSILOXANE DOW CORNING TORAY CO., LTD. (JP) 2006-12-28 WO disclosed