SCHEMBL5264877

SCHEMBL5264877

Cc1ccc(C#Cc2ccc(-c3nc4ccccn4c3NC(C)(C)C)s2)nc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1B P35368 1/20 0.48
MAPT P10636 3/20 0.48
PKM P14618 3/20 0.48
PKLR P30613 2/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
GAA P10253 4/20 0.43
TP53 P04637 1/20 0.43
TOP2A P11388 1/20 0.42
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
GFER P55789 1/20 0.42
BRD4 O60885 1/20 0.42
TRIM24 O15164 1/20 0.42
SALL4 Q9UJQ4 1/20 0.42
TRIM33 Q9UPN9 1/20 0.42
BACE1 P56817 6/20 0.40
BACE2 Q9Y5Z0 6/20 0.40
HDAC4 P56524 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
HDAC9 Q9UKV0 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5129281 0.99 ADRA1B (0.47) ADRA1BMAPTPKMPKLRSMN1; SMN2
SCHEMBL5315271 0.88 BRD4 (0.44) ADRA1BMAPTPKMPKLRSMN1; SMN2
SCHEMBL5118071 0.87 ADRA1B (0.51) ADRA1BMAPTPKMPKLRSMN1; SMN2
Hydrochloric Acid SCHEMBL5127004 0.87 BRD4 (0.44) ADRA1BMAPTPKMPKLRSMN1; SMN2
Hydrochloric Acid SCHEMBL5116906 0.87 ADRA1B (0.50) ADRA1BMAPTPKMPKLRSMN1; SMN2
Hydrochloric Acid SCHEMBL5127777 0.87 ADRA1B (0.50) ADRA1BMAPTPKMPKLRSMN1; SMN2
SCHEMBL5263543 0.83 ADRA1B (0.53) ADRA1BMAPTPKMPKLRSMN1; SMN2
Hydrochloric Acid SCHEMBL5121300 0.83 ADRA1B (0.50) ADRA1BMAPTPKMPKLRSMN1; SMN2
Hydrochloric Acid SCHEMBL5129005 0.82 ADRA1B (0.52) ADRA1BMAPTPKMPKLRSMN1; SMN2
SCHEMBL5128705 0.82 PKM (0.55) ADRA1BMAPTPKMPKLRSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1791840-A1 SUBSTITUTED BICYCLIC IMIDAZO-3-YLAMINE COMPOUNDS Grünenthal GmbH (DE) 2007-06-06 EP disclosed
WO-2006029980-A1 SUBSTITUTED BICYCLIC IMIDAZO-3-YLAMINE COMPOUNDS Grünenthal GmbH (DE) 2006-03-23 WO disclosed