SCHEMBL5265181

SCHEMBL5265181

CCOC(=O)C(Br)C1CCNCC1

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 7/20 0.47
SLC6A3 Q01959 7/20 0.47
SLC6A4 P31645 6/20 0.47
CPN1 P15169 1/20 0.40
CPB2 Q96IY4 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.39
SMYD3 Q9H7B4 1/20 0.39
MAPT P10636 1/20 0.35
PKM P14618 1/20 0.35
ALDH1A1 P00352 2/20 0.33
OPRD1 P41143 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL381187 0.87 L3MBTL1 (0.44) L3MBTL1ALDH1A1NPSR1
SCHEMBL21009822 0.87 L3MBTL1 (0.44) L3MBTL1ALDH1A1NPSR1
SCHEMBL17200481 0.83 ALDH1A1 (0.45) SLC6A2SLC6A3SLC6A4L3MBTL1ALDH1A1
SCHEMBL28249755 0.83 L3MBTL1 (0.42) L3MBTL1ALDH1A1NPSR1
SCHEMBL31547138 0.83 ALDH1A1 (0.45) SLC6A2SLC6A3SLC6A4L3MBTL1ALDH1A1
SCHEMBL197612 0.81 ALDH1A1 (0.48) L3MBTL1ALDH1A1NPSR1
SCHEMBL198506 0.81 ALDH1A1 (0.48) L3MBTL1ALDH1A1NPSR1
SCHEMBL5268464 0.81 SLC6A2 (0.44) SLC6A2SLC6A3SLC6A4CPN1CPB2
SCHEMBL11395732 0.81 L3MBTL1 (0.53) SLC6A2SLC6A3SLC6A4CPN1CPB2
SCHEMBL2254747 0.80 SLC6A2 (0.48) SLC6A2SLC6A3SLC6A4CPN1CPB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3096754-A1 METALLO-BETA-LACTAMASE INHIBITORS Merck Sharp & Dohme Corp. (US) 2016-11-30 EP disclosed
WO-2015112441-A1 METALLO-BETA-LACTAMASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2015-07-30 WO disclosed
EP-1802602-A1 SUBSTITUTED DIPIPERDINE CCR2 ANTAGONISTS JANSSEN PHARMACEUTICA N.V. (BE) 2007-07-04 EP disclosed
WO-2006036527-A1 SUBSTITUTED DIPIPERDINE CCR2 ANTAGONISTS JANSSEN PHARMACEUTICA, N.V. (BE) 2006-04-06 WO disclosed