SCHEMBL5266344

SCHEMBL5266344

CC(C)(C)Nc1c(-c2ccc(C#Cc3cccc(S(N)(=O)=O)c3)s2)nc2ccccn12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1B P35368 1/20 0.44
TOP2A P11388 1/20 0.41
TRIM24 O15164 1/20 0.41
SALL4 Q9UJQ4 1/20 0.41
TRIM33 Q9UPN9 1/20 0.41
CA12 O43570 4/20 0.40
CA1 P00915 4/20 0.40
CA2 P00918 4/20 0.40
CA9 Q16790 4/20 0.40
BACE1 P56817 5/20 0.40
BACE2 Q9Y5Z0 5/20 0.40
HDAC7 Q8WUI4 2/20 0.38
HDAC9 Q9UKV0 2/20 0.38
HDAC5 Q9UQL6 2/20 0.38
HDAC3 O15379 1/20 0.38
NCOR2 Q9Y618 1/20 0.38
MAPT P10636 2/20 0.38
GAA P10253 2/20 0.38
PKM P14618 2/20 0.38
TP53 P04637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5118578 0.99 ADRA1B (0.44) ADRA1BTOP2ATRIM24SALL4TRIM33
SCHEMBL5264250 0.87 ADRA1B (0.48) ADRA1BTOP2ATRIM24SALL4TRIM33
Hydrochloric Acid SCHEMBL5116930 0.86 ADRA1B (0.47) ADRA1BTOP2ATRIM24SALL4TRIM33
SCHEMBL5113916 0.85 ADRA1B (0.44) ADRA1BTOP2ATRIM24SALL4TRIM33
SCHEMBL5117968 0.85 ADRA1B (0.48) ADRA1BTOP2ATRIM24SALL4TRIM33
SCHEMBL5117557 0.85 ADRA1B (0.48) ADRA1BTOP2ATRIM24SALL4TRIM33
SCHEMBL5266397 0.84 TOP2A (0.48) ADRA1BTOP2ATRIM24SALL4TRIM33
Hydrochloric Acid SCHEMBL5128215 0.84 TOP2A (0.47) ADRA1BTOP2ATRIM24SALL4TRIM33
SCHEMBL5114390 0.83 TOP2A (0.56) ADRA1BTOP2ATRIM24SALL4TRIM33
Hydrochloric Acid SCHEMBL5128015 0.83 TOP2A (0.48) ADRA1BTOP2ATRIM24SALL4TRIM33

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1791840-A1 SUBSTITUTED BICYCLIC IMIDAZO-3-YLAMINE COMPOUNDS Grünenthal GmbH (DE) 2007-06-06 EP claimed
WO-2006029980-A1 SUBSTITUTED BICYCLIC IMIDAZO-3-YLAMINE COMPOUNDS Grünenthal GmbH (DE) 2006-03-23 WO claimed
EP-1791840-A1 SUBSTITUTED BICYCLIC IMIDAZO-3-YLAMINE COMPOUNDS Grünenthal GmbH (DE) 2007-06-06 EP disclosed
WO-2006029980-A1 SUBSTITUTED BICYCLIC IMIDAZO-3-YLAMINE COMPOUNDS Grünenthal GmbH (DE) 2006-03-23 WO disclosed