SCHEMBL5266502

SCHEMBL5266502

CC(=O)Nc1cccc(C(=O)Nc2c[nH]nc2C(=O)NCc2ccccc2)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.56
L3MBTL1 Q9Y468 1/20 0.56
KMT2A Q03164 2/20 0.50
MEN1 O00255 1/20 0.50
LMNA P02545 2/20 0.49
MAPK1 P28482 2/20 0.49
RAB9A P51151 2/20 0.49
PTGIR P43119 1/20 0.48
ALPL P05186 1/20 0.48
ALPI P09923 1/20 0.48
ALPG P10696 1/20 0.48
HPGD P15428 1/20 0.48
HTT P42858 1/20 0.48
CLK1 P49759 1/20 0.47
CDK14 O94921 3/20 0.47
CCNY Q8ND76 3/20 0.47
CHRM3 P20309 1/20 0.47
ITGA4 P13612 1/20 0.47
ITGB7 P26010 1/20 0.47
NPC1 O15118 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5270190 0.90 LMNA (0.53) ALDH1A1L3MBTL1KMT2AMEN1LMNA
SCHEMBL4287309 0.88 CDK14 (0.47) ALDH1A1L3MBTL1KMT2AMEN1RAB9A
SCHEMBL5271991 0.87 CDK14 (0.55) KMT2AMEN1RAB9AALPLALPI
SCHEMBL5274230 0.86 HPGD (0.49) ALDH1A1KMT2AMAPK1HPGDITGA4
SCHEMBL4293189 0.85 MAPT (0.51) KMT2AMEN1RAB9AHPGDNPC1
SCHEMBL5266768 0.85 CLK1 (0.52) ALDH1A1KMT2AMEN1RAB9AALPL
SCHEMBL4292708 0.84 CDK14 (0.48) RAB9AALPLALPIALPGCLK1
SCHEMBL4284373 0.84 CDK14 (0.48) ALDH1A1KMT2AMEN1RAB9AALPL
SCHEMBL5266452 0.84 NPC1 (0.57) ALDH1A1L3MBTL1KMT2AMEN1LMNA
SCHEMBL5269902 0.84 CLK1 (0.51) ALDH1A1KMT2AMEN1RAB9AALPL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1847531-A1 PYRAZOLE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2007-10-24 EP disclosed