SCHEMBL5269902

SCHEMBL5269902

CNC(=O)c1n[nH]cc1NC(=O)c1cccc(NC(C)=O)c1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CLK1 P49759 1/20 0.51
CDK14 O94921 5/20 0.50
CCNY Q8ND76 5/20 0.50
TSHR P16473 1/20 0.49
ALPL P05186 1/20 0.48
ALPI P09923 1/20 0.48
ALPG P10696 1/20 0.48
POLB P06746 4/20 0.46
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
ALDH1A1 P00352 2/20 0.44
RAB9A P51151 2/20 0.44
NPC1 O15118 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5271991 0.89 CDK14 (0.55) CLK1CDK14CCNYTSHRALPL
SCHEMBL5266768 0.89 CLK1 (0.52) CLK1CDK14CCNYTSHRALPL
SCHEMBL5269232 0.88 CLK1 (0.49) CLK1CDK14CCNYTSHRALPL
SCHEMBL4284373 0.85 CDK14 (0.48) CLK1CDK14CCNYTSHRALPL
SCHEMBL4292708 0.85 CDK14 (0.48) CLK1CDK14CCNYTSHRALPL
SCHEMBL5266502 0.84 ALDH1A1 (0.56) CLK1CDK14CCNYALPLALPI
SCHEMBL5271516 0.84 SMYD3 (0.55) CLK1CDK14CCNYTSHRALPL
SCHEMBL4283610 0.84 CDK14 (0.49) CLK1CDK14CCNYTSHRALPL
SCHEMBL4287309 0.84 CDK14 (0.47) CLK1CDK14CCNYTSHRALPL
SCHEMBL4289521 0.83 CDK14 (0.53) CLK1CDK14CCNYTSHRALPL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1847531-A1 PYRAZOLE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2007-10-24 EP disclosed