Hydroxyamine

Hydroxyamine

SCHEMBL5266580

COc1cc(C(=O)N2CC[C@@H]2C(=O)O)cc(Br)c1OC.NO

nearest known ligand 0.52

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.52
APOBEC3A P31941 1/20 0.52
HTT P42858 1/20 0.52
APOBEC3G Q9HC16 1/20 0.52
KMT2A Q03164 3/20 0.48
GAA P10253 1/20 0.45
ALDH1A1 P00352 5/20 0.44
CYP1A2 P05177 1/20 0.44
TUBB4A P04350 1/20 0.43
TUBB P07437 1/20 0.43
TUBA3C P0DPH7 1/20 0.43
TUBA1B P68363 1/20 0.43
TUBA4A P68366 1/20 0.43
TUBB4B P68371 1/20 0.43
TUBB3 Q13509 1/20 0.43
TUBB2A Q13885 1/20 0.43
TUBB8 Q3ZCM7 1/20 0.43
TUBA3E Q6PEY2 1/20 0.43
TUBA1A Q71U36 1/20 0.43
TUBA1C Q9BQE3 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydroxyamine SCHEMBL5266577 1.00 TSHR (0.52) TSHRAPOBEC3AHTTAPOBEC3GKMT2A
Hydroxyamine SCHEMBL5274861 0.91 GAA (0.53) KMT2AGAAALDH1A1CYP1A2POLB
Hydroxyamine SCHEMBL5274854 0.91 GAA (0.53) KMT2AGAAALDH1A1CYP1A2POLB
SCHEMBL3546824 0.87 FKBP1A (0.55) TSHRAPOBEC3AHTTAPOBEC3GKMT2A
SCHEMBL3546826 0.87 FKBP1A (0.55) TSHRAPOBEC3AHTTAPOBEC3GKMT2A
SCHEMBL3544922 0.86 TSHR (0.49) TSHRAPOBEC3AHTTAPOBEC3GKMT2A
SCHEMBL3544921 0.86 TSHR (0.49) TSHRAPOBEC3AHTTAPOBEC3GKMT2A
SCHEMBL11998537 0.81 FKBP1A (0.56) KMT2AGAAALDH1A1CYP1A2POLB
SCHEMBL3554498 0.79 ALDH1A1 (0.48) TSHRAPOBEC3AHTTAPOBEC3GKMT2A
SCHEMBL3554500 0.79 ALDH1A1 (0.48) TSHRAPOBEC3AHTTAPOBEC3GKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539744-A4 N-HYDROXYAMIDE DERIVATIVES POSSESSING ANTIBACTERIAL ACTIVITY VICURON PHARM INC (US) 2007-06-06 EP disclosed
EP-1539744-A2 N-HYDROXYAMIDE DERIVATIVES POSSESSING ANTIBACTERIAL ACTIVITY Vicuron Pharmaceuticals, Inc. (US) 2005-06-15 EP disclosed
WO-2004007444-A2 N-HYDROXYAMIDE DERIVATIVES POSSESSING ANTIBACTERIAL ACTIVITY VICURON PHARMACEUTICALS, INC. (US) 2004-01-22 WO disclosed