SCHEMBL5267116

SCHEMBL5267116

Cc1cn2c(Nc3cc(C)[nH]n3)nc(-c3ccc4c(c3)[N]C(=O)N4)cc2n1

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GSK3A P49840 2/20 0.36
GSK3B P49841 2/20 0.36
AURKA O14965 8/20 0.34
AURKB Q96GD4 8/20 0.34
SYK P43405 5/20 0.33
ITK Q08881 1/20 0.31
IGF1R P08069 1/20 0.31
FLT4 P35916 1/20 0.30
KDR P35968 1/20 0.30
RET P07949 1/20 0.30
SRC P12931 1/20 0.30
EIF2AK2 P19525 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3042602 0.82 GSK3A (0.38) GSK3AGSK3BAURKAAURKBSYK
SCHEMBL13221325 0.81 GSK3B (0.54) GSK3AGSK3BAURKAAURKBITK
SCHEMBL13221349 0.79 GSK3B (0.43) GSK3AGSK3BAURKAAURKBSRC
SCHEMBL13221315 0.77 GSK3A (0.41) GSK3AGSK3BAURKAAURKBSYK
SCHEMBL3031628 0.76 GSK3A (0.42) GSK3AGSK3BAURKAAURKBITK
SCHEMBL13221341 0.76 ALDH1A1 (0.46) GSK3AGSK3BAURKAAURKBSRC
SCHEMBL5262600 0.75 GSK3A (0.41) GSK3AGSK3BAURKAAURKBITK
SCHEMBL3037557 0.75 GSK3A (0.39) GSK3AGSK3BAURKAAURKBSYK
SCHEMBL5262598 0.75 NPC1 (0.41) GSK3AGSK3BAURKAAURKBITK
SCHEMBL3037823 0.75 HTR6 (0.37) GSK3AGSK3BAURKBSYKIGF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1812439-A2 KINASE INHIBITORS Takeda San Diego, Inc. (US) 2007-08-01 EP disclosed
WO-2006044687-A2 KINASE INHIBITORS TAKEDA SAN DIEGO, INC. (US) 2006-04-27 WO disclosed