SCHEMBL5267196

SCHEMBL5267196

O=c1cc(-c2ccc(OC3CCNCC3)cc2)ccn1C(F)F

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.48
PTGS2 P35354 6/20 0.46
HRH1 P35367 2/20 0.42
ROCK1 Q13464 3/20 0.40
ROCK2 O75116 1/20 0.40
PRKACA P17612 1/20 0.40
PRKCD Q05655 1/20 0.40
PRKG1 Q13976 1/20 0.40
PKN1 Q16512 1/20 0.40
PKN2 Q16513 1/20 0.40
AAK1 Q2M2I8 1/20 0.40
CDC42BPA Q5VT25 1/20 0.40
Q6ZSR9 Q6ZSR9 1/20 0.40
BMP2K Q9NSY1 1/20 0.40
CDC42BPB Q9Y5S2 1/20 0.40
TLR9 Q9NR96 1/20 0.40
TLR8 Q9NR97 1/20 0.40
TLR7 Q9NYK1 1/20 0.40
KHK P50053 1/20 0.40
ALOX5 P09917 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2116740 0.83 HRH3 (0.48) HRH3PTGS2KCNH2
SCHEMBL2114205 0.81 HRH3 (0.52) HRH3KCNH2
SCHEMBL2114120 0.81 HRH3 (0.54) HRH3KCNH2
SCHEMBL2019376 0.75 HRH1 (0.70) HRH3HRH1ROCK1ROCK2PRKACA
SCHEMBL14431595 0.71 HRH1 (0.59) HRH3HRH1
SCHEMBL12975670 0.71 QDPR (0.41) PTGS2ALOX5PTGS1
SCHEMBL2115508 0.70 HRH3 (0.63) HRH3HRH1ROCK1ROCK2PRKACA
SCHEMBL2117437 0.70 HRH3 (0.54) HRH3KCNH2
SCHEMBL18322912 0.69 HRH3 (0.44) HRH3HRH1ROCK1TLR9TLR8
SCHEMBL5204218 0.69 HRH1 (0.79) HRH3HRH1ROCK1KHKGRK6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1820797-A1 SUBSTITUTED PYRIDONE DERIVATIVE BANYU PHARMACEUTICAL CO., LTD. (JP) 2007-08-22 EP disclosed