SCHEMBL5269293

SCHEMBL5269293

CC(C)NC(=O)c1n[nH]cc1NS(=O)(=O)c1cc(Cl)ccc1Cl

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 5/20 0.50
HPGD P15428 1/20 0.49
TSHR P16473 1/20 0.49
ACLY P53396 2/20 0.45
MAPK1 P28482 1/20 0.44
ALPL P05186 1/20 0.43
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
POLB P06746 1/20 0.42
MAPT P10636 2/20 0.42
HTT P42858 2/20 0.42
BRD4 O60885 2/20 0.42
HSD11B1 P28845 1/20 0.42
ALDH1A1 P00352 2/20 0.42
LMNA P02545 2/20 0.42
TDP1 Q9NUW8 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
NHERF1 O14745 1/20 0.42
PIK3CD O00329 1/20 0.41
PIK3CA P42336 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5270409 0.89 MCL1 (0.52) MCL1HPGDTSHRACLYMAPK1
SCHEMBL5271647 0.83 MCL1 (0.46) MCL1HPGDTSHRACLYMAPK1
SCHEMBL5270643 0.83 MEN1 (0.55) MCL1HPGDTSHRACLYMAPK1
SCHEMBL5265851 0.81 MCL1 (0.48) MCL1HPGDTSHRACLYMAPK1
SCHEMBL5271640 0.80 KCNA5 (0.51) MCL1HPGDTSHRACLYMAPK1
SCHEMBL5268776 0.79 CCKAR (0.52) MCL1HPGDTSHRACLYMEN1
SCHEMBL5269115 0.77 HPGD (0.48) HPGDMAPK1MEN1KMT2APOLB
SCHEMBL5265268 0.76 KCNA5 (0.46) HPGDTSHRMEN1KMT2APOLB
SCHEMBL5270919 0.76 KCNA5 (0.51) MCL1TSHRMEN1KMT2AHTT
SCHEMBL5271810 0.75 KCNA5 (0.50) TSHRPOLBMAPTALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1847531-A1 PYRAZOLE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2007-10-24 EP disclosed