SCHEMBL5273255

SCHEMBL5273255

CC(=O)Nc1cccc(C(=O)Nc2c[nH]nc2C(=O)N2CCCC2)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRD O14764 1/20 0.50
GABRA1 P14867 1/20 0.50
GABRB1 P18505 1/20 0.50
GABRA5 P31644 1/20 0.50
GABRA3 P34903 1/20 0.50
GABRA2 P47869 1/20 0.50
GABRB2 P47870 1/20 0.50
GABRA4 P48169 1/20 0.50
POLB P06746 1/20 0.48
TP53 P04637 2/20 0.48
ALDH1A1 P00352 1/20 0.48
HPGD P15428 1/20 0.48
HTT P42858 1/20 0.48
KDM4E B2RXH2 1/20 0.48
GAA P10253 1/20 0.47
ATM Q13315 1/20 0.46
ALPL P05186 1/20 0.46
ALPI P09923 1/20 0.46
ALPG P10696 1/20 0.46
CLK1 P49759 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5266768 0.83 CLK1 (0.52) POLBALDH1A1HTTALPLALPI
SCHEMBL5271504 0.83 HPGD (0.53) POLBALDH1A1HPGDGAAKMT2A
SCHEMBL5269232 0.83 CLK1 (0.49) POLBALPLALPIALPGCLK1
SCHEMBL5269902 0.82 CLK1 (0.51) POLBALDH1A1ALPLALPIALPG
SCHEMBL5269043 0.82 KMT2A (0.41) POLBALDH1A1HPGDKDM4EGAA
SCHEMBL5271991 0.81 CDK14 (0.55) POLBALPLALPIALPGCLK1
SCHEMBL5271516 0.80 SMYD3 (0.55) POLBHPGDALPLALPIALPG
SCHEMBL18478351 0.78 HPGD (0.69) GABRDGABRA1GABRB1GABRA5GABRA3
SCHEMBL4284373 0.77 CDK14 (0.48) POLBALDH1A1KDM4EALPLALPI
SCHEMBL4292708 0.77 CDK14 (0.48) POLBKDM4EALPLALPIALPG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1847531-A1 PYRAZOLE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2007-10-24 EP disclosed