SCHEMBL5269232

SCHEMBL5269232

CC(=O)Nc1cccc(C(=O)Nc2c[nH]nc2C(=O)NC(C)C)c1

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CLK1 P49759 1/20 0.49
CDK14 O94921 4/20 0.49
CCNY Q8ND76 4/20 0.49
ROCK2 O75116 2/20 0.48
PKM P14618 1/20 0.47
TSHR P16473 1/20 0.47
ALPL P05186 1/20 0.47
ALPI P09923 1/20 0.47
ALPG P10696 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP3A5 P20815 1/20 0.47
POLB P06746 2/20 0.44
ADRB2 P07550 1/20 0.43
ADRB1 P08588 1/20 0.43
ADRB3 P13945 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5266768 0.90 CLK1 (0.52) CLK1CDK14CCNYTSHRALPL
SCHEMBL5269902 0.88 CLK1 (0.51) CLK1CDK14CCNYTSHRALPL
SCHEMBL5271991 0.87 CDK14 (0.55) CLK1CDK14CCNYTSHRALPL
SCHEMBL4293839 0.84 PAX8 (0.59) CLK1CDK14CCNYTSHRALPL
SCHEMBL5271516 0.84 SMYD3 (0.55) CLK1CDK14CCNYPKMTSHR
SCHEMBL5267481 0.83 MDM4 (0.49) PKMPOLBMEN1KMT2A
SCHEMBL4283194 0.83 PAX8 (0.65) CLK1CDK14CCNYTSHRPOLB
SCHEMBL5273255 0.83 GABRD (0.50) CLK1CDK14CCNYTSHRALPL
SCHEMBL4284373 0.83 CDK14 (0.48) CLK1CDK14CCNYTSHRALPL
SCHEMBL4292708 0.83 CDK14 (0.48) CLK1CDK14CCNYPKMTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1847531-A1 PYRAZOLE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2007-10-24 EP disclosed