SCHEMBL5276352

SCHEMBL5276352

O=C(O)Oc1cn([C@H]2C[C@H]2F)c2c(Cl)c(N3CCN(CCOCCO)CC3)c(F)cc2c1=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.41
POLB P06746 2/20 0.41
CHRM2 P08172 1/20 0.41
CHRM1 P11229 1/20 0.41
OPRM1 P35372 1/20 0.41
OPRD1 P41143 1/20 0.41
BCL2A1 Q16548 1/20 0.36
KDM4E B2RXH2 4/20 0.35
LMNA P02545 1/20 0.34
NSD2 O96028 1/20 0.34
PABPC1 P11940 1/20 0.34
CASP6 P55212 1/20 0.34
PAX8 Q06710 1/20 0.34
HPGD P15428 2/20 0.34
HSD17B10 Q99714 2/20 0.34
HRH3 Q9Y5N1 2/20 0.34
ALB P02768 1/20 0.34
TUBB4A P04350 1/20 0.34
TUBB P07437 1/20 0.34
TUBA3C P0DPH7 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5179509 1.00 ALDH1A1 (0.41) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL967206 0.90 ALDH1A1 (0.51) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL966606 0.90 ALDH1A1 (0.51) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL967204 0.90 ALDH1A1 (0.51) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL5178871 0.90 ALDH1A1 (0.49) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL5277216 0.89 KCNH2 (0.42) ALDH1A1POLBOPRM1KDM4ELMNA
SCHEMBL5282151 0.86 KDM4E (0.46) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL5280465 0.85 EPHX2 (0.36) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL5280454 0.85 EPHX2 (0.36) ALDH1A1POLBCHRM2CHRM1OPRM1
SCHEMBL5279342 0.85 EPHX2 (0.36) ALDH1A1POLBCHRM2CHRM1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1768973-B1 SUBSTITUTED QUINOLONES AICURIS GMBH & CO KG (DE) 2007-12-05 EP disclosed