SCHEMBL527853

SCHEMBL527853

O=c1[nH]cnc2c(F)cc(S(=O)(=O)Cl)cc12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IP6K1 Q92551 7/20 0.51
PARP1 P09874 9/20 0.50
BCL2 P10415 1/20 0.46
MCL1 Q07820 1/20 0.46
IGF1R P08069 2/20 0.40
PIM1 P11309 2/20 0.40
CLK2 P49760 2/20 0.40
GSK3A P49840 2/20 0.40
GSK3B P49841 2/20 0.40
DYRK1A Q13627 2/20 0.40
CLK4 Q9HAZ1 2/20 0.40
AURKA O14965 1/20 0.40
DAPK3 O43293 1/20 0.40
JAK2 O60674 1/20 0.40
PRKD3 O94806 1/20 0.40
MAP4K4 O95819 1/20 0.40
PAK4 O96013 1/20 0.40
ABL1 P00519 1/20 0.40
CSF1R P07333 1/20 0.40
RET P07949 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18128478 0.78 IP6K1 (0.56) IP6K1PARP1BCL2MCL1IGF1R
SCHEMBL525865 0.75 PARP1 (0.49) IP6K1PARP1PIM1ALDH1A1PIM2
SCHEMBL18130618 0.74 IP6K1 (0.56) IP6K1PARP1BCL2MCL1IGF1R
SCHEMBL3659063 0.72 PARP1 (0.61) IP6K1PARP1PIM1ACVR1ALDH1A1
SCHEMBL8568798 0.69 PARP1 (0.61) IP6K1PARP1BCL2MCL1IGF1R
SCHEMBL526730 0.67 PARP1 (1.00) IP6K1PARP1BCL2MCL1IGF1R
SCHEMBL527342 0.66 PGR (0.34) PARP1ALDH1A1
SCHEMBL15846231 0.65 IP6K1 (0.48) IP6K1PARP1BCL2MCL1MAP4K4
SCHEMBL12068369 0.65 PARP1 (0.51) IP6K1PARP1BCL2MCL1IGF1R
SCHEMBL31559173 0.65 PARP1 (0.47) IP6K1PARP1BCL2MCL1IGF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012014109-A1 HETEROCYCLIC SULFONAMIDES AS INHIBITORS OF TRANSFER RNA SYNTHETASE FOR USE AS ANTIBACTERIAL AGENTS RANBAXY LABORATORIES LIMITED (IN) 2012-02-02 WO disclosed