SCHEMBL5280111

SCHEMBL5280111

O=C(NCCOC(=O)N(c1ccccc1-c1ccccc1)N1CC[CH]CC1)c1ccc(CN2CCC(CO)CC2)s1

nearest known ligand 0.37

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 11/20 0.37
POLB P06746 1/20 0.36
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
SLC2A1 P11166 1/20 0.34
ACKR3 P25106 2/20 0.34
HTR7 P34969 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5276784 0.90 EPHX2 (0.37) EPHX2SLC2A1ACKR3HTR7
SCHEMBL5276039 0.80 PDCD1 (0.33) HTR7
SCHEMBL6027281 0.79 PDCD1 (0.37) ACKR3
SCHEMBL2639950 0.76 CHRM2 (0.37) POLBKDM4EALDH1A1
SCHEMBL5281205 0.76 ACKR3 (0.32) ACKR3
SCHEMBL5272613 0.75 PDCD1 (0.38) POLBALDH1A1
SCHEMBL5722183 0.73 HPGD (0.40) ALDH1A1
SCHEMBL4694436 0.73 NPC1 (0.38) ALDH1A1
SCHEMBL4695640 0.72 PDCD1 (0.34) ACKR3
SCHEMBL2639688 0.72 POLB (0.44) EPHX2POLBKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1856112-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS Theravance, Inc. (US) 2007-11-21 EP claimed
WO-2006099032-A1 BIPHENYL COMPOUNDS USEFUL AS MUSCARINIC RECEPTOR ANTAGONISTS THERAVANCE, INC. (US) 2006-09-21 WO claimed