SCHEMBL5280451

SCHEMBL5280451

COC(=O)/C=C/c1cccc(C2OCCO2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.49
KDM4E B2RXH2 4/20 0.49
TTR P02766 1/20 0.48
APP P05067 1/20 0.48
PTPN1 P18031 1/20 0.46
PRKDC P78527 1/20 0.45
EPHX2 P34913 1/20 0.45
SIRT2 Q8IXJ6 1/20 0.44
SIRT1 Q96EB6 1/20 0.44
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
TYR P14679 1/20 0.44
CA7 P43166 1/20 0.44
CA9 Q16790 1/20 0.44
CA14 Q9ULX7 1/20 0.44
MAPT P10636 2/20 0.44
GLA P06280 1/20 0.44
THRB P10828 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5280456 1.00 ALDH1A1 (0.49) ALDH1A1KDM4ETTRAPPPTPN1
SCHEMBL8803514 0.85 GLA (0.49) ALDH1A1KDM4EAPPMAPTGLA
SCHEMBL69618 0.79 TTR (0.66) ALDH1A1KDM4ETTRAPPPTPN1
SCHEMBL3065424 0.75 CA12 (0.66) ALDH1A1KDM4ETTRAPPPTPN1
SCHEMBL30676338 0.75 CA12 (0.66) ALDH1A1KDM4ETTRAPPPTPN1
SCHEMBL2631340 0.75 CA12 (0.66) ALDH1A1KDM4ETTRAPPPTPN1
SCHEMBL2169771 0.74 NR1H4 (0.44) ALDH1A1KDM4ETTRAPPPTPN1
SCHEMBL3413478 0.74 NR1H4 (0.46) ALDH1A1KDM4ETTRAPPPTPN1
SCHEMBL2614742 0.73 TTR (0.58) ALDH1A1KDM4ETTRAPPPTPN1
SCHEMBL4084338 0.73 TTR (0.58) ALDH1A1KDM4ETTRAPPPTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1313560-B1 CATALYST FOR AROMATIC C-O, C-N, and C-C BOND FORMATION UNIV YALE (US) 2007-12-19 EP disclosed
EP-1313560-A4 CATALYST FOR AROMATIC C-O, C-N, and C-C BOND FORMATION UNIV YALE (US) 2005-02-09 EP disclosed
EP-1313560-A1 CATALYST FOR AROMATIC C-O, C-N, and C-C BOND FORMATION YALE UNIVERSITY (US) 2003-05-28 EP disclosed
US-6562989-B2 Bicyclopentyl iron ligand and transition metal catalyst YALE UNIVERSITY 2003-05-13 US disclosed
US-20030008768-A1 Catalyst for aromatic C-O, C-N, and C-C bond formation NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2003-01-09 US disclosed
WO-2002011883-A1 CATALYST FOR AROMATIC C-O, C-N, and C-C BOND FORMATION YALE UNIVERSITY (US) 2002-02-14 WO disclosed