SCHEMBL5280924

SCHEMBL5280924

CC(C)(C)OC(=O)N(CCc1ccc(OCc2ccccc2)cc1)S(=O)(=O)c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTB4R Q15722 1/20 0.51
LTB4R2 Q9NPC1 1/20 0.51
PTGES O14684 2/20 0.50
KCNH2 Q12809 1/20 0.50
ALOX5 P09917 4/20 0.49
KEAP1 Q14145 1/20 0.48
FFAR1 O14842 1/20 0.47
FFAR4 Q5NUL3 1/20 0.47
POLB P06746 2/20 0.47
LMNA P02545 1/20 0.47
MAPT P10636 1/20 0.47
HTT P42858 1/20 0.47
BCL2 P10415 1/20 0.46
MMP2 P08253 2/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
MMP9 P14780 1/20 0.45
CA9 Q16790 1/20 0.45
ADAMTS4 O75173 1/20 0.44
MMP13 P45452 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3014165 0.82 LTB4R (0.67) LTB4RLTB4R2ALOX5FFAR1FFAR4
SCHEMBL14229905 0.81 LTB4R (0.56) LTB4RLTB4R2ALOX5FFAR1FFAR4
SCHEMBL4453600 0.80 LTB4R (0.55) LTB4RLTB4R2ALOX5FFAR1FFAR4
SCHEMBL4449671 0.80 LTB4R (0.55) LTB4RLTB4R2ALOX5FFAR1FFAR4
SCHEMBL9533718 0.79 LTB4R (0.54) LTB4RLTB4R2ALOX5FFAR1FFAR4
SCHEMBL4450404 0.79 BCHE (0.55) LTB4RLTB4R2ALOX5FFAR1FFAR4
SCHEMBL4880111 0.78 CA12 (0.45) ALOX5POLBLMNAMAPTHTT
SCHEMBL4453618 0.77 BCHE (0.52) LTB4RLTB4R2ALOX5FFAR1FFAR4
SCHEMBL7835952 0.77 LTB4R (0.52) LTB4RLTB4R2ALOX5FFAR1FFAR4
SCHEMBL7063146 0.77 STAT5B (0.47) PTGESPOLBCA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1851208-A1 MACROCYCLIC COMPOUNDS USEFUL AS BACE INHIBITORS Novartis AG (CH) 2007-11-07 EP disclosed
WO-2006074950-A1 MACROCYCLIC COMPOUNDS USEFUL AS BACE INHIBITORS NOVARTIS AG (CH) 2006-07-20 WO disclosed