SCHEMBL5281026

SCHEMBL5281026

COC(=O)c1ccc(C2C(O)CN(C(=O)O)CC2O[Si](C(C)C)(C(C)C)C(C)C)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 6/20 0.36
HSD17B10 Q99714 5/20 0.36
ALDH1A1 P00352 5/20 0.36
KDM4E B2RXH2 4/20 0.36
HPGD P15428 3/20 0.36
GAA P10253 2/20 0.36
CASP1 P29466 2/20 0.36
CASP7 P55210 2/20 0.36
ATM Q13315 2/20 0.36
GRIN2B Q13224 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
MAPK1 P28482 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
NAMPT P43490 1/20 0.33
GLA P06280 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2684431 1.00 TSHR (0.36) TSHRHSD17B10ALDH1A1KDM4EHPGD
SCHEMBL3905395 0.87 PAX8 (0.36) TSHRALDH1A1HPGDSMN1; SMN2MEN1
SCHEMBL2344278 0.85 NPC1 (0.41) ALDH1A1SMN1; SMN2MEN1KMT2ANPC1
SCHEMBL3908901 0.82
SCHEMBL3943583 0.81 KDM4E (0.34) ALDH1A1KDM4ESMN1; SMN2MEN1KMT2A
SCHEMBL2685066 0.79 DRD2 (0.37)
SCHEMBL2683683 0.79 MAPT (0.41) TSHRHSD17B10ALDH1A1HPGDGAA
SCHEMBL2682948 0.79 KDM4E (0.39) TSHRHSD17B10ALDH1A1KDM4EHPGD
SCHEMBL5280813 0.79 KDM4E (0.39) TSHRHSD17B10ALDH1A1KDM4EHPGD
SCHEMBL3912312 0.78

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1863763-A1 3,4,5-SUBSTITUTED PIPERIDINES AS RENIN INHIBITORS Speedel Experimenta AG (CH) 2007-12-12 EP disclosed
WO-2006103275-A1 3,4,5-SUBSTITUTED PIPERIDINES AS RENIN INHIBITORS SPEEDEL EXPERIMENTA AG (CH) 2006-10-05 WO disclosed