SCHEMBL5281640

SCHEMBL5281640

CC(O)CCc1ccccc1Br

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 3/20 0.50
TYR P14679 2/20 0.46
IDO1 P14902 2/20 0.39
GPR52 Q9Y2T5 1/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
SLC6A3 Q01959 1/20 0.39
TSHR P16473 2/20 0.38
HPGD P15428 1/20 0.37
ANPEP P15144 1/20 0.37
PYCR1 P32322 1/20 0.36
RIPK1 Q13546 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14036598 0.89 TAAR1 (0.47) TAAR1TYRIDO1GPR52TSHR
SCHEMBL15532115 0.85 TAAR1 (0.47) TAAR1IDO1GPR52SLC6A2SLC6A4
SCHEMBL4365156 0.83 TAAR1 (0.54) TAAR1IDO1GPR52SLC6A2SLC6A4
SCHEMBL30521500 0.80 SLC6A2 (0.61) TAAR1IDO1GPR52SLC6A2SLC6A4
SCHEMBL623814 0.80 SLC6A2 (0.61) TAAR1IDO1GPR52SLC6A2SLC6A4
SCHEMBL14997308 0.79 TAAR1 (0.44) TAAR1IDO1SLC6A2SLC6A4TSHR
SCHEMBL15319327 0.79 TAAR1 (0.44) TAAR1IDO1SLC6A2SLC6A4TSHR
SCHEMBL625240 0.79 TAAR1 (0.44) TAAR1IDO1SLC6A2SLC6A4TSHR
SCHEMBL29679614 0.79 TAAR1 (0.44) TAAR1IDO1SLC6A2SLC6A4TSHR
SCHEMBL17593488 0.78 TAAR1 (0.48) TAAR1IDO1GPR52TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2834233-A1 NEW ALPHA2 ADRENOCEPTOR AGONISTS Orion Corporation (FI) 2015-02-11 EP disclosed
WO-2013150173-A1 NEW ALPHA2 ADRENOCEPTOR AGONISTS ORION CORPORATION (FI) 2013-10-10 WO disclosed
EP-1313560-B1 CATALYST FOR AROMATIC C-O, C-N, and C-C BOND FORMATION UNIV YALE (US) 2007-12-19 EP disclosed
EP-1313560-A4 CATALYST FOR AROMATIC C-O, C-N, and C-C BOND FORMATION UNIV YALE (US) 2005-02-09 EP disclosed
EP-1313560-A1 CATALYST FOR AROMATIC C-O, C-N, and C-C BOND FORMATION YALE UNIVERSITY (US) 2003-05-28 EP disclosed
US-6562989-B2 Bicyclopentyl iron ligand and transition metal catalyst YALE UNIVERSITY 2003-05-13 US disclosed
US-20030008768-A1 Catalyst for aromatic C-O, C-N, and C-C bond formation NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2003-01-09 US disclosed
WO-2002011883-A1 CATALYST FOR AROMATIC C-O, C-N, and C-C BOND FORMATION YALE UNIVERSITY (US) 2002-02-14 WO disclosed