SCHEMBL5281653

SCHEMBL5281653

COc1ccc(N2CCCCC2)cc1Nc1ncc(Br)c([AsH]c2ccccc2S(=O)(=O)NC(C)C)n1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 8/20 0.52
EGFR P00533 3/20 0.52
PLK4 O00444 2/20 0.52
LCK P06239 2/20 0.52
FYN P06241 2/20 0.52
IGF1R P08069 2/20 0.52
EPHA2 P29317 2/20 0.52
FLT3 P36888 2/20 0.52
LIMK1 P53667 2/20 0.52
PTK2 Q05397 2/20 0.52
PTK6 Q13882 2/20 0.52
PTK2B Q14289 2/20 0.52
AURKB Q96GD4 2/20 0.52
PRKD2 Q9BZL6 2/20 0.52
SLK Q9H2G2 2/20 0.52
CDC7 O00311 1/20 0.52
CHEK1 O14757 1/20 0.52
AURKA O14965 1/20 0.52
DCLK1 O15075 1/20 0.52
PDPK1 O15530 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4093702 0.85 ALK (0.70) ALKEGFRPLK4LCKFYN
SCHEMBL4089503 0.79 ALK (0.70) ALKEGFRPLK4LCKFYN
SCHEMBL4100115 0.79 ALK (0.63) ALKEGFRPLK4LCKFYN
SCHEMBL4095865 0.79 ULK1 (0.74) ALKEGFRPLK4LCKFYN
SCHEMBL4089370 0.78 ALK (0.68) ALKEGFRPLK4LCKFYN
SCHEMBL4095269 0.77 ALK (0.81) ALKEGFRPLK4LCKFYN
SCHEMBL4096592 0.75 ZAP70 (0.78) ALKEGFRPLK4LCKFYN
SCHEMBL5290384 0.75 ZAP70 (0.53) ALKEGFRPLK4LCKFYN
SCHEMBL4100866 0.75 ALK (0.66) ALKEGFRPLK4LCKFYN
SCHEMBL4103561 0.74 ULK1 (0.67) ALKEGFRPLK4LCKFYN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1784392-A2 PYRIMIDINE DERIVATIVES Novartis AG (CH) 2007-05-16 EP claimed
WO-2006021454-A2 PYRIMIDINE DERIVATIVES NOVARTIS AG (CH) 2006-03-02 WO claimed