SCHEMBL5284520

SCHEMBL5284520

CC1CCN(C(=O)c2ccc(N)c(N3CCN(C)CC3)c2)c2ccccc2N1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2C P18825 1/20 0.42
KDM4E B2RXH2 4/20 0.41
HSD17B10 Q99714 2/20 0.41
ALDH1A1 P00352 1/20 0.41
GAA P10253 3/20 0.40
MAPK1 P28482 2/20 0.40
MAPT P10636 1/20 0.40
HTT P42858 1/20 0.40
RECQL P46063 1/20 0.40
PTK2B Q14289 1/20 0.40
BRD4 O60885 3/20 0.39
POLB P06746 3/20 0.38
LMNA P02545 1/20 0.36
CRBN Q96SW2 2/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
USP2 O75604 1/20 0.36
AVPR1A P37288 2/20 0.36
CREBBP Q92793 1/20 0.36
OXTR P30559 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4912725 1.00 ADRA2C (0.42) ADRA2CKDM4EHSD17B10ALDH1A1GAA
SCHEMBL4904747 0.88 BRD4 (0.39) KDM4EALDH1A1MAPK1MAPTBRD4
SCHEMBL4912161 0.85 ALDH1A1 (0.46) ALDH1A1GAAMAPK1MAPTHTT
SCHEMBL4915013 0.79 MAP3K11 (0.41) CREBBPOXTR
SCHEMBL4902302 0.78 TSHR (0.41) ALDH1A1MAPK1MAPTHTTBRD4
SCHEMBL4909211 0.77 BRD4 (0.35) ALDH1A1MAPK1MAPTBRD4LMNA
SCHEMBL4902490 0.76 AVPR2 (0.50) KDM4EALDH1A1HTTLMNAMEN1
SCHEMBL4912334 0.76 GPBAR1 (0.42) ALDH1A1MAPK1MAPTHTTBRD4
SCHEMBL4907240 0.76 GPBAR1 (0.42) ALDH1A1MAPK1MAPTHTTBRD4
SCHEMBL4906946 0.74 GPBAR1 (0.41) ALDH1A1MAPK1MAPTHTTBRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1820799-A1 2,3,4,5-TETRAHYDRO-1H-1,5-BENZODIAZEPINE DERIVATIVE AND MEDICINAL COMPOSITION Wakamoto Pharmaceutical Co., Ltd. (JP) 2007-08-22 EP disclosed