Pyridine

Pyridine

SCHEMBL528579

[Cl-].[Cl-].[Pd+2].c1ccncc1.c1ccncc1.c1ccncc1.c1ccncc1

nearest known ligand 0.90

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEBDKRB2CHRM1CHRM2CHRM3CHRNA1CHRNB1CHRNDCHRNECHRNGGUCY1A1GUCY1A2GUCY1B1GUCY1B2NAMPTPTAFRSLC10A2SLC6A2SLC6A3TACR1dacAdacBdacCftsImrcAmrcBmrdA

The experimentally established mechanism targets of Pyridine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SLC6A2 known ✓ P23975 1/20 0.33
SLC6A3 known ✓ Q01959 1/20 0.33
TSHR P16473 2/20 0.90
NAPRT Q6XQN6 1/20 0.90
TDP1 Q9NUW8 1/20 0.90
NOTUM Q6P988 1/20 0.39
SLC6A4 P31645 1/20 0.33
ALDH1A1 P00352 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2A6 P11509 1/20 0.32
LMNA P02545 1/20 0.31
MAPT P10636 1/20 0.31
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
TP53 P04637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pyridine SCHEMBL29404917 1.00
Pyridine SCHEMBL11313895 1.00
Pyridine SCHEMBL4950936 1.00 TSHR (0.90) TSHRNAPRTTDP1NOTUMSLC6A2
SCHEMBL3052767 0.95 TSHR (1.00) TSHRNAPRTTDP1NOTUMSLC6A2
Pyridine SCHEMBL180431 0.95 TSHR (1.00) TSHRNAPRTTDP1NOTUMSLC6A2
Pyridine SCHEMBL16 0.95
Pyridine SCHEMBL933604 0.95 TSHR (1.00) TSHRNAPRTTDP1NOTUMSLC6A2
Pyridine SCHEMBL1654468 0.95
Pyridine SCHEMBL9037865 0.95 TSHR (1.00) TSHRNAPRTTDP1NOTUMSLC6A2
Benzene SCHEMBL1261317 0.95 TSHR (1.00) TSHRNAPRTTDP1NOTUMSLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 25 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210340285-A1 METHOD FOR PRODUCING HYDROGENATED NITRILE RUBBER AND HNBR COMPOSITIONS THEREOF ARLANXEO DEUTSCHLAND GMBH (DE) 2021-11-04 US claimed
EP-3827029-A1 METHOD FOR PRODUCING HYDROGENATED NITRILE RUBBER AND HNBR COMPOSITIONS THEREOF ARLANXEO Deutschland GmbH (DE) 2021-06-02 EP claimed
WO-2020020677-A1 METHOD FOR PRODUCING HYDROGENATED NITRILE RUBBER AND HNBR COMPOSITIONS THEREOF ARLANXEO DEUTSCHLAND GMBH (DE) 2020-01-30 WO claimed
US-20210340285-A1 METHOD FOR PRODUCING HYDROGENATED NITRILE RUBBER AND HNBR COMPOSITIONS THEREOF ARLANXEO DEUTSCHLAND GMBH (DE) 2021-11-04 US disclosed
EP-3827029-A1 METHOD FOR PRODUCING HYDROGENATED NITRILE RUBBER AND HNBR COMPOSITIONS THEREOF ARLANXEO Deutschland GmbH (DE) 2021-06-02 EP disclosed
US-10781270-B2 Method of production of highly saturated nitrile rubber ZEON CORPORATION (JP) 2020-09-22 US disclosed
WO-2020020677-A1 METHOD FOR PRODUCING HYDROGENATED NITRILE RUBBER AND HNBR COMPOSITIONS THEREOF ARLANXEO DEUTSCHLAND GMBH (DE) 2020-01-30 WO disclosed
EP-3252084-B1 METHOD FOR PRODUCING HIGHLY SATURATED NITRILE RUBBER ZEON CORP (JP) 2019-08-28 EP disclosed
US-20180016360-A1 METHOD OF PRODUCTION OF HIGHLY SATURATED NITRILE RUBBER ZEON CORPORATION (JP) 2018-01-18 US disclosed
EP-3252084-A1 METHOD FOR PRODUCING HIGHLY SATURATED NITRILE RUBBER Zeon Corporation (JP) 2017-12-06 EP disclosed
EP-2598537-B1 HYDROGENATION OF DIENE-BASED POLYMERS ARLANXEO DEUTSCHLAND GMBH (DE) 2017-05-03 EP disclosed
WO-2012013697-A2 HYDROGENATION OF DIENE-BASED POLYMERS LANXESS DEUTSCHLAND GMBH (DE) 2012-02-02 WO disclosed
US-7923514-B2 such as acrylonitrile-butadiene copolymer, using as hydrogenation catalyst a platinum group metal or its compound, and a basic compound ZEON CORPORATION (JP) 2011-04-12 US disclosed
EP-1454924-B1 METHOD OF HYDROGENATING CONJUGATED DIENE POLYMER, HYDROGENATION CATALYST SYSTEM, AND COMPOSITION OF BASIC CONJUGATED DIENE POLYMER ZEON CORP (JP) 2009-03-18 EP disclosed
US-20080132649-A1 METHOD OF HYDROGENATING CONJUGATED DIENE POLYMER, HYDROGENATION CATALYST SYSTEM, AND COMPOSTION OF BASIC, CONJUGATED DIENE POLYMER ZEON CORPORATION 2008-06-05 US disclosed
US-20040242800-A1 Method of hydrogenating conjugated diene polymer, hydrogenation catalyst system, and composition of basic conjugated diene polymer ZEON CORPORATION (JP) 2004-12-02 US disclosed
EP-1454924-A1 METHOD OF HYDROGENATING CONJUGATED DIENE POLYMER, HYDROGENATION CATALYST SYSTEM, AND COMPOSITION OF BASIC CONJUGATED DIENE POLYMER Zeon Corporation (JP) 2004-09-08 EP disclosed
US-5169901-A Catalyzing in presence of high molecular complex of palladium compound and a nitrile grop-containing polymer NIPPON ZEON CO., LTD. (JP) 1992-12-08 US disclosed
US-5164457-A Palladium catalyst NIPPON ZEON CO., LTD. (JP) 1992-11-17 US disclosed
US-5128297-A Catalysis with palladium compound and acrylonitrile-conjugated diene polymer complex NIPPON ZEON CO., LTD. (JP) 1992-07-07 US disclosed