SCHEMBL5286249

SCHEMBL5286249

O=[N+]([O-])c1ccc([N]CC(F)(F)F)cc1C(F)(F)F

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT6 Q8N6T7 1/20 0.50
AR P10275 9/20 0.43
CYP3A4 P08684 3/20 0.43
LMNA P02545 2/20 0.43
CYP1A2 P05177 2/20 0.43
CYP2C9 P11712 2/20 0.43
TSHR P16473 2/20 0.43
CYP2C19 P33261 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
PGR P06401 2/20 0.43
CES2 O00748 1/20 0.43
ABCB11 O95342 1/20 0.43
ALDH1A1 P00352 1/20 0.43
GLA P06280 1/20 0.43
ADORA3 P0DMS8 1/20 0.43
CHRM1 P11229 1/20 0.43
ALOX15 P16050 1/20 0.43
TBXA2R P21731 1/20 0.43
AADAC P22760 1/20 0.43
MAPK1 P28482 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14048317 0.81 SIRT6 (0.48) SIRT6ARCYP3A4LMNACYP1A2
SCHEMBL332231 0.77 SIRT6 (0.45) SIRT6ARCYP3A4LMNACYP1A2
SCHEMBL3925839 0.76 SIRT6 (0.44) SIRT6ARCYP3A4LMNACYP1A2
SCHEMBL7569166 0.75 AR (0.45) SIRT6ARCYP3A4LMNACYP1A2
SCHEMBL12972551 0.75 AR (0.45) SIRT6ARCYP3A4LMNACYP1A2
SCHEMBL1998640 0.72 CYP3A4 (0.52) SIRT6ARCYP3A4LMNACYP1A2
SCHEMBL31138869 0.72 ALDH1A1 (0.53) SIRT6ARCYP3A4LMNACYP1A2
SCHEMBL29788520 0.72 ATM (0.60) SIRT6ARCYP3A4LMNACYP1A2
SCHEMBL2639009 0.72 SIRT6 (0.51) SIRT6ARCYP3A4LMNACYP1A2
SCHEMBL377777 0.72 ATM (0.60) SIRT6ARCYP3A4LMNACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007005887-A2 ANDROGEN RECEPTOR MODULATOR COMPOUNDS, COMPOSITIONS AND USES THEREOF LIGAND PHARMACEUTICALS INCORPORATED (US) 2007-01-11 WO disclosed