SCHEMBL5286981

SCHEMBL5286981

COc1cccc(-c2cccc3ccccc23)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.55
GPR84 Q9NQS5 1/20 0.53
CYP1A2 P05177 9/20 0.51
CYP2C9 P11712 6/20 0.51
CYP3A4 P08684 5/20 0.51
CYP2B6 P20813 5/20 0.51
CYP2D6 P10635 4/20 0.51
AHR P35869 3/20 0.51
NR1I3 Q14994 3/20 0.51
CYP2C19 P33261 3/20 0.51
VDR P11473 2/20 0.51
CYP11B1 P15538 1/20 0.51
CYP11B2 P19099 1/20 0.51
CYP1A1 P04798 3/20 0.51
CYP1B1 Q16678 3/20 0.51
ADORA2A P29274 2/20 0.50
ALOX5 P09917 1/20 0.50
ADORA1 P30542 1/20 0.49
CLK4 Q9HAZ1 2/20 0.48
NR1I2 O75469 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27651329 0.88 BRD4 (0.46) BRD4GPR84CYP1A2CYP2C9CYP3A4
SCHEMBL2020140 0.85 ABL1 (0.59) BRD4CYP1A2CYP2C9CYP3A4CYP2B6
SCHEMBL9538506 0.84 GPR84 (0.59) BRD4GPR84CYP1A2CYP2C9CYP3A4
SCHEMBL13241142 0.83 GPR84 (0.52) BRD4GPR84CYP1A2CYP2C9CYP3A4
SCHEMBL13241136 0.83 MAOB (0.56) BRD4GPR84CYP1A2CYP2C9CYP3A4
Methyl Alcohol SCHEMBL29235314 0.83 CYP11B1 (0.65) CYP1A2CYP2C9CYP3A4CYP2B6CYP2D6
SCHEMBL13241148 0.83 MAOB (0.52) BRD4GPR84CYP1A2CYP2C9CYP3A4
SCHEMBL14134369 0.83 CYP1A2 (0.50) BRD4GPR84CYP1A2CYP2C9CYP3A4
SCHEMBL312278 0.82 KMT2A (0.56) BRD4GPR84CYP1A2CYP2C9CYP3A4
SCHEMBL13241129 0.82 BRD4 (0.51) BRD4CYP1A2CYP2C9CYP3A4CYP2B6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102958892-A Method for preparing chemical compounds of interest by aromatic nucleophilic substitution CENTRE NAT RECH SCIENT 2013-03-06 CN disclosed
EP-1313560-B1 CATALYST FOR AROMATIC C-O, C-N, and C-C BOND FORMATION UNIV YALE (US) 2007-12-19 EP disclosed
EP-1313560-A4 CATALYST FOR AROMATIC C-O, C-N, and C-C BOND FORMATION UNIV YALE (US) 2005-02-09 EP disclosed
EP-1313560-A1 CATALYST FOR AROMATIC C-O, C-N, and C-C BOND FORMATION YALE UNIVERSITY (US) 2003-05-28 EP disclosed
US-6562989-B2 Bicyclopentyl iron ligand and transition metal catalyst YALE UNIVERSITY 2003-05-13 US disclosed
US-20030008768-A1 Catalyst for aromatic C-O, C-N, and C-C bond formation NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2003-01-09 US disclosed
WO-2002011883-A1 CATALYST FOR AROMATIC C-O, C-N, and C-C BOND FORMATION YALE UNIVERSITY (US) 2002-02-14 WO disclosed
EP-0532531-A1 PHENOL AND PYRIDINOL DERIVATIVES AS PHARMACEUTICALS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1993-03-24 EP disclosed
WO-1991017987-A1 PHENOL AND PYRIDINOL DERIVATIVES AS PHARMACEUTICALS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1991-11-28 WO disclosed