SCHEMBL528913

SCHEMBL528913

CCCCc1cnc2ccc(Br)cc2c1O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.45
NFKB1 P19838 2/20 0.45
RAB9A P51151 2/20 0.45
NFKB2 Q00653 2/20 0.45
RELA Q04206 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
GAA P10253 2/20 0.45
HTT P42858 5/20 0.43
CCNC P24863 1/20 0.43
CDK8 P49336 1/20 0.43
TSHR P16473 1/20 0.41
LMNA P02545 3/20 0.40
ALDH1A1 P00352 1/20 0.40
ALK Q9UM73 1/20 0.39
ATM Q13315 1/20 0.38
MAPK1 P28482 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
MAPT P10636 2/20 0.37
TYR P14679 1/20 0.37
EIF4A1 P60842 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL529732 0.91 HTT (0.44) NPC1NFKB1RAB9ANFKB2RELA
SCHEMBL529341 0.83 CYP1A2 (0.46) NPC1NFKB1RAB9ANFKB2RELA
SCHEMBL528924 0.82 HTT (0.40) SMN1; SMN2GAAHTTCCNCCDK8
SCHEMBL8413790 0.80 RARB (0.44) NPC1NFKB1RAB9ANFKB2RELA
SCHEMBL7850047 0.79 TLR7 (0.43) SMN1; SMN2GAALMNAALDH1A1MAPK1
SCHEMBL529735 0.78 HTT (0.42) SMN1; SMN2GAAHTTCCNCCDK8
SCHEMBL27448960 0.76 HTT (0.38) GAAHTTTSHRLMNAALDH1A1
SCHEMBL529947 0.75 HTT (0.39) SMN1; SMN2GAAHTTCCNCCDK8
SCHEMBL6529277 0.75 TLR7 (0.48) SMN1; SMN2GAALMNAALDH1A1ATM
SCHEMBL529322 0.74 CYP1A2 (0.48) NPC1SMN1; SMN2GAAHTTCCNC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2597955-A1 QUINOLINE DERIVATIVES AND MELK INHIBITORS CONTAINING THE SAME OncoTherapy Science, Inc. (JP) 2013-06-05 EP disclosed
WO-2012016082-A1 QUINOLINE DERIVATIVES AND MELK INHIBITORS CONTAINING THE SAME ONCOTHERAPY SCIENCE, INC. (JP) 2012-02-02 WO disclosed