SCHEMBL529947

SCHEMBL529947

O=CCc1cnc2ccc(Br)cc2c1O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 6/20 0.39
TSHR P16473 1/20 0.39
CHEK1 O14757 1/20 0.39
PIM1 P11309 1/20 0.39
AKT1 P31749 1/20 0.39
FLT3 P36888 1/20 0.39
PIM3 Q86V86 1/20 0.39
LMNA P02545 3/20 0.38
MAPT P10636 1/20 0.38
ALDH1A1 P00352 2/20 0.37
ALK Q9UM73 1/20 0.37
KDM4E B2RXH2 1/20 0.37
HPGD P15428 1/20 0.37
MTOR P42345 1/20 0.37
NCOA1 Q15788 1/20 0.37
NCOA3 Q9Y6Q9 1/20 0.37
ERN1 O75460 1/20 0.37
GABRA1 P14867 1/20 0.36
GABRG2 P18507 1/20 0.36
GABRB3 P28472 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL529686 0.82 CYP1A2 (0.40) HTTTSHRCHEK1PIM1AKT1
SCHEMBL27448960 0.80 HTT (0.38) HTTTSHRCHEK1PIM1AKT1
SCHEMBL529732 0.78 HTT (0.44) HTTTSHRCHEK1PIM1AKT1
SCHEMBL529735 0.77 HTT (0.42) HTTTSHRCHEK1PIM1AKT1
SCHEMBL528913 0.75 NPC1 (0.45) HTTTSHRLMNAMAPTALDH1A1
SCHEMBL528924 0.74 HTT (0.40) HTTTSHRCHEK1PIM1AKT1
SCHEMBL16589027 0.74 ALK (0.44) HTTTSHRCHEK1PIM1AKT1
SCHEMBL17598440 0.73 HTT (0.42) HTTTSHRCHEK1PIM1AKT1
SCHEMBL17578990 0.73 ALK (0.43) HTTTSHRCHEK1PIM1AKT1
SCHEMBL14899564 0.71 TNF (0.45) HTTTSHRCHEK1PIM1AKT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2597955-A1 QUINOLINE DERIVATIVES AND MELK INHIBITORS CONTAINING THE SAME OncoTherapy Science, Inc. (JP) 2013-06-05 EP disclosed
WO-2012016082-A1 QUINOLINE DERIVATIVES AND MELK INHIBITORS CONTAINING THE SAME ONCOTHERAPY SCIENCE, INC. (JP) 2012-02-02 WO disclosed