SCHEMBL528924

SCHEMBL528924

CC(C)CCc1cnc2ccc(Br)cc2c1O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 5/20 0.40
LMNA P02545 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
MAPT P10636 2/20 0.40
NPSR1 Q6W5P4 2/20 0.38
RXFP1 Q9HBX9 2/20 0.38
GAA P10253 1/20 0.38
TSHR P16473 2/20 0.38
MCL1 Q07820 1/20 0.37
ALDH1A1 P00352 2/20 0.37
CCNC P24863 2/20 0.36
CDK8 P49336 2/20 0.36
ALK Q9UM73 1/20 0.35
MAPK1 P28482 1/20 0.35
PRNP P04156 1/20 0.35
MAPK10 P53779 1/20 0.35
CHEK1 O14757 1/20 0.34
PIM1 P11309 1/20 0.34
AKT1 P31749 1/20 0.34
FLT3 P36888 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL529735 0.86 HTT (0.42) HTTLMNASMN1; SMN2MAPTNPSR1
SCHEMBL529732 0.84 HTT (0.44) HTTLMNASMN1; SMN2MAPTNPSR1
SCHEMBL528765 0.83 RXFP1 (0.42) HTTLMNASMN1; SMN2MAPTNPSR1
SCHEMBL528913 0.82 NPC1 (0.45) HTTLMNASMN1; SMN2MAPTNPSR1
SCHEMBL27448960 0.75 HTT (0.38) HTTLMNAMAPTNPSR1RXFP1
SCHEMBL529947 0.74 HTT (0.39) HTTLMNASMN1; SMN2MAPTNPSR1
SCHEMBL15191355 0.73 HTT (0.50) HTTLMNASMN1; SMN2NPSR1RXFP1
SCHEMBL15191291 0.73 HTT (0.47) HTTLMNASMN1; SMN2MAPTNPSR1
SCHEMBL14899564 0.72 TNF (0.45) HTTLMNASMN1; SMN2MAPTNPSR1
SCHEMBL16589027 0.72 ALK (0.44) HTTLMNASMN1; SMN2MAPTTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2597955-A1 QUINOLINE DERIVATIVES AND MELK INHIBITORS CONTAINING THE SAME OncoTherapy Science, Inc. (JP) 2013-06-05 EP disclosed
WO-2012016082-A1 QUINOLINE DERIVATIVES AND MELK INHIBITORS CONTAINING THE SAME ONCOTHERAPY SCIENCE, INC. (JP) 2012-02-02 WO disclosed