SCHEMBL5289461

SCHEMBL5289461

Cc1cc(C)cc(C)c1.O=S(=O)=NO

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.43
TPMT P51580 1/20 0.42
TSHR P16473 3/20 0.38
CYP3A4 P08684 2/20 0.36
CYP1A2 P05177 1/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA3 P07451 1/20 0.36
CA4 P22748 1/20 0.36
CA6 P23280 1/20 0.36
CA5A P35218 1/20 0.36
CA7 P43166 1/20 0.36
CA9 Q16790 1/20 0.36
CA13 Q8N1Q1 1/20 0.36
CA14 Q9ULX7 1/20 0.36
CA5B Q9Y2D0 1/20 0.36
ACHE P22303 2/20 0.35
SELL P14151 1/20 0.35
SELP P16109 1/20 0.35
SELE P16581 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27507877 0.77 ALDH1A1 (0.50) ALDH1A1TPMTTSHRCYP3A4CA1
SCHEMBL29212116 0.77 ALDH1A1 (0.45) ALDH1A1TPMTTSHRCYP3A4CYP1A2
Toluene SCHEMBL28569928 0.76 LMNA (0.55) ALDH1A1TSHRACHEHPGD
SCHEMBL296587 0.73
Benzene SCHEMBL28169481 0.70
Methyl Alcohol SCHEMBL28397318 0.69 ALDH1A1 (0.64) ALDH1A1TPMTTSHRCYP3A4ACHE
Hydrochloric Acid SCHEMBL28239385 0.69
SCHEMBL28425258 0.69 ALDH1A1 (0.57) ALDH1A1TPMTTSHRCYP3A4CA1
SCHEMBL19376983 0.69 ALDH1A1 (0.57) ALDH1A1TPMTTSHRCYP3A4CA1
Methyl Alcohol SCHEMBL27974355 0.69 ALDH1A1 (0.64) ALDH1A1TPMTTSHRCYP3A4ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 25 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112724133-B Preparation method of 6-bromopyrazolo [1,5-a ] pyridine 湖南复瑞生物医药技术有限责任公司 2022-03-25 CN claimed
CN-112724133-A Preparation method of 6-bromopyrazolo [1,5-a ] pyridine 湖南复瑞生物医药技术有限责任公司 2021-04-30 CN claimed
JP-57048966-A None JP disclosed
CN-113788790-A Aromatic heterocyclic amide derivative and application thereof 华东理工大学 2021-12-14 CN disclosed
CN-106008369-B The bicyclic dihydropyrimidinonesand being substituted and its purposes as the active inhibitor of Neutrophil elastase 勃林格殷格翰国际有限公司 2019-06-21 CN disclosed
CN-106045920-B The bicyclic dihydropyrimidinonesand being substituted and its purposes as the active inhibitor of Neutrophil elastase 勃林格殷格翰国际有限公司 2018-10-19 CN disclosed
CN-106045921-B The bicyclic dihydropyrimidinonesand being substituted and its purposes as the active inhibitor of Neutrophil elastase 勃林格殷格翰国际有限公司 2018-09-25 CN disclosed
CN-105722839-B Pesticidally active bicyclic heterocycles with sulphur-containing substituents 先正达参股股份有限公司 2018-04-06 CN disclosed
CN-104995186-B Substituted bicyclic dihydropyrimidinones and their use as inhibitors of neutrophil elastase activity 勃林格殷格翰国际有限公司 2017-06-20 CN disclosed
CN-103333102-B Pyridyl-N-cyano sulfo oxime compound and preparation method thereof BEIJING GREENCHEM TECHNOLOGY CO LTD 2015-06-17 CN disclosed
CN-104447591-A Energetic compound 3,3'-diamido-2,2'-2(2,2,2-trinitroethyl)-5,5'-linked triazole-diamine and preparation method and intermediate thereof INST CHEMICAL MATERIAL CHINA ACADEMY ENGINEERING PHYSICS 2015-03-25 CN disclosed
EP-0604920-A1 Novel cephalosporin compounds LUCKY LTD. (KR) 1994-07-06 EP disclosed
US-4612311-A ANXIOLYTIC AGENTS WARNER-LAMBERT COMPANY (US) 1986-09-16 US disclosed
JP-S5748966-A PYRIDYLSULFOXYIMINES WAKO PURE CHEM IND LTD 1982-03-20 JP disclosed
US-4259494-A ANTIHISTAMINIC, ANTITUSSIVE, ANTIINFLAMMATORY, SEDATIVE, DIURETIC WARNER-LAMBERT COMPANY (US) 1981-03-31 US disclosed
US-4110448-A ANTIHISTAMINE, ANTITUSSIVE, ANTIINFLAMMATORY, SEDATIVE, DIURETIC WARNER-LAMBERT COMPANY (US) 1978-08-29 US disclosed
US-4076723-A ANTIHISTAMINES, ANTITUSSIVE AGENTS, ANTIINFLAMMATORY AGENTS, SEDATIVES, DIURETICS WARNER-LAMBERT COMPANY (US) 1978-02-28 US disclosed
US-4033981-A ANTIHISTOMINIC, ANTIINFLAMMATORY, SEDATIVES, DIURETICS WARNER-LAMBERT COMPANY (US) 1977-07-05 US disclosed
US-3992376-A ANTIHISTAMINES, ANTITUSSIVES, SEDATIVES, ANTIINFLAMMATORY AGENTS AND DIURETICS WARNER-LAMBERT COMPANY (US) 1976-11-16 US disclosed
US-3978052-A ANTIHISTAMINIC, ANTITUSSIVE, ANTIINFLAMMATORY, DIURETIC WARNER-LAMBERT COMPANY (US) 1976-08-31 US disclosed