SCHEMBL529063

SCHEMBL529063

CN(C)CCNc1ccc(Nc2c(CC=O)cnc3ccc(Br)cc23)cn1

nearest known ligand 0.50

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MELK Q14680 8/20 0.50
EGFR P00533 9/20 0.44
ERBB2 P04626 1/20 0.36
FLT3 P36888 1/20 0.36
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
GAA P10253 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL529522 0.84 MELK (0.51) MELKEGFRERBB2
SCHEMBL529001 0.83 MELK (0.74) MELK
SCHEMBL529912 0.83 MELK (0.48) MELKEGFRERBB2FLT3KDM4E
SCHEMBL530051 0.83 MELK (0.47) MELKEGFRERBB2
SCHEMBL529062 0.82 MELK (0.71) MELKEGFRKDM4EMEN1GAA
SCHEMBL529716 0.81 MELK (0.46) MELK
SCHEMBL529572 0.80 MELK (0.76) MELK
SCHEMBL529700 0.79 MELK (0.73) MELK
SCHEMBL12504780 0.76 EGFR (0.47) MELKEGFRFLT3
SCHEMBL529723 0.74 MELK (0.49) MELKEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2597955-A1 QUINOLINE DERIVATIVES AND MELK INHIBITORS CONTAINING THE SAME OncoTherapy Science, Inc. (JP) 2013-06-05 EP disclosed
WO-2012016082-A1 QUINOLINE DERIVATIVES AND MELK INHIBITORS CONTAINING THE SAME ONCOTHERAPY SCIENCE, INC. (JP) 2012-02-02 WO disclosed