SCHEMBL529522

SCHEMBL529522

CN(C)CCOc1ccc(Nc2c(CC=O)cnc3ccc(Br)cc23)cn1

nearest known ligand 0.51

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MELK Q14680 14/20 0.51
EGFR P00533 3/20 0.39
ATM Q13315 2/20 0.37
ERBB2 P04626 2/20 0.37
CSF1R P07333 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL529063 0.84 MELK (0.50) MELKEGFRERBB2
SCHEMBL530051 0.83 MELK (0.47) MELKEGFRERBB2
Hydrochloric Acid SCHEMBL12505070 0.83 MELK (0.72) MELKATM
SCHEMBL529521 0.82 MELK (0.72) MELK
SCHEMBL529716 0.81 MELK (0.46) MELK
SCHEMBL15130443 0.80 MELK (0.53) MELKATM
SCHEMBL530043 0.79 MELK (0.74) MELK
SCHEMBL17434850 0.76 MELK (0.78) MELKATM
SCHEMBL17434914 0.76 MELK (0.79) MELK
SCHEMBL12504771 0.75 MELK (0.46) MELKEGFRATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2597955-A1 QUINOLINE DERIVATIVES AND MELK INHIBITORS CONTAINING THE SAME OncoTherapy Science, Inc. (JP) 2013-06-05 EP disclosed
WO-2012016082-A1 QUINOLINE DERIVATIVES AND MELK INHIBITORS CONTAINING THE SAME ONCOTHERAPY SCIENCE, INC. (JP) 2012-02-02 WO disclosed