SCHEMBL530051

SCHEMBL530051

CN(C)CCc1ccc(Nc2c(CC=O)cnc3ccc(Br)cc23)cc1

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MELK Q14680 15/20 0.47
TAAR1 Q96RJ0 1/20 0.39
NPC1 O15118 1/20 0.39
NCOA1 Q15788 1/20 0.39
NCOA3 Q9Y6Q9 1/20 0.39
EGFR P00533 2/20 0.38
ERBB2 P04626 1/20 0.38
WEE1 P30291 1/20 0.37
KCNH2 Q12809 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL529716 0.90 MELK (0.46) MELK
SCHEMBL529522 0.83 MELK (0.51) MELKEGFRERBB2
SCHEMBL529063 0.83 MELK (0.50) MELKEGFRERBB2
SCHEMBL5655413 0.82 MELK (0.48) MELKTAAR1NPC1NCOA1NCOA3
SCHEMBL529048 0.82 MELK (0.73) MELK
SCHEMBL530050 0.81 MELK (0.69) MELK
SCHEMBL529513 0.79 MELK (0.48) MELK
SCHEMBL528701 0.79 MELK (0.74) MELK
SCHEMBL529029 0.78 MELK (0.71) MELK
SCHEMBL529164 0.77 MELK (0.75) MELK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2597955-A1 QUINOLINE DERIVATIVES AND MELK INHIBITORS CONTAINING THE SAME OncoTherapy Science, Inc. (JP) 2013-06-05 EP disclosed
WO-2012016082-A1 QUINOLINE DERIVATIVES AND MELK INHIBITORS CONTAINING THE SAME ONCOTHERAPY SCIENCE, INC. (JP) 2012-02-02 WO disclosed