SCHEMBL529065

SCHEMBL529065

Cc1ccc(C(=O)NCCCCCC(=O)Nc2ccccc2N)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 18/20 1.00
HDAC1 Q13547 15/20 1.00
HDAC2 Q92769 2/20 1.00
NCOR2 Q9Y618 2/20 1.00
HDAC8 Q9BY41 1/20 1.00
HDAC4 P56524 1/20 0.79

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1938496 1.00 HDAC3 (1.00) HDAC3HDAC1HDAC2NCOR2HDAC8
SCHEMBL31060469 1.00 HDAC3 (1.00) HDAC3HDAC1HDAC2NCOR2HDAC8
SCHEMBL1937829 0.99 HDAC3 (0.98) HDAC3HDAC1HDAC2NCOR2HDAC8
SCHEMBL1938110 0.88 HDAC3 (1.00) HDAC3HDAC1HDAC2NCOR2HDAC8
SCHEMBL1938122 0.88 HDAC3 (1.00) HDAC3HDAC1HDAC2NCOR2HDAC8
SCHEMBL1938221 0.88 HDAC3 (1.00) HDAC3HDAC1HDAC2NCOR2HDAC8
SCHEMBL1937223 0.88 HDAC3 (1.00) HDAC3HDAC1HDAC2NCOR2HDAC8
SCHEMBL16011065 0.88 HDAC4 (1.00) HDAC3HDAC1HDAC2NCOR2HDAC8
SCHEMBL1937932 0.88 HDAC3 (1.00) HDAC3HDAC1HDAC2NCOR2HDAC8
SCHEMBL1937980 0.88 HDAC1 (1.00) HDAC3HDAC1HDAC2NCOR2HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 402 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026107052-A1 COMBINATION TREATMENTS USING EPIGENETIC INHIBITION AND SYNGRI-MEDIATED FRATAXIN EXPRESSION ST. JUDE CHILDREN'S RESEARCH HOSPITAL, INC. (US) 2026-05-21 WO claimed
US-20260125650-A1 METHODS AND COMPOSITIONS FOR GENERATING HEPATOCYTES TRAILHEAD BIOSYSTEMS INC (US) 2026-05-07 US claimed
EP-4720316-A2 NON-VIRAL CELL ENGINEERING Arsenal Biosciences, Inc. (US) 2026-04-08 EP claimed
US-20250268948-A1 COMPOSITIONS AND METHODS FOR TREATING POST ACUTE SEQUELAE OF SARS-COV-2 INFECTION (LONG COVID) AE CAPITAL LIMITED (VG) 2025-08-28 US claimed
US-20250205286-A1 COMPOSITIONS, REAGENTS, AND METHODS FOR TREATING PITT-HOPKINS SYNDROME AE CAPITAL LIMITED (VG) 2025-06-26 US claimed
US-20250188422-A1 INDUCED TOTIPOTENT POTENTIAL STEM CELLS, METHODS OF MAKING AND USING PEKING UNIVERSITY (CN) 2025-06-12 US claimed
US-20250161243-A1 MEF2 TRANSCRIPTIONAL ACTIVATORS TO TREAT NEUROLOGIC CONDITIONS THE SCRIPPS RESEARCH INSTITUTE 2025-05-22 US claimed
US-20250144056-A1 ANTIMICROBIAL HOST DEFENSE PEPTIDE-INDUCING COMPOSITIONS AND METHODS OF PRODUCTION AND USE THEREOF BOARD OF REGENTS FOR THE OKLAHOMA AGRICULTURAL AND MECH COLLEGES (US) 2025-05-08 US claimed
US-20250115871-A1 METHODS TO IMPROVE ENDURING HEMATOPOIETIC STEM CELL TRANSPLANTATION TRAILHEAD BIOSYSTEMS INC. 2025-04-10 US claimed
WO-2025059442-A1 MODULATING PLANT RESPONSES TO STRESS AND GROWTH WITH CHEMICALS REMOTE EPIGENETICS INC. (US) 2025-03-20 WO claimed
US-20170231931-A1 PRODUCTS FOR THE TREATMENT AND PREVENTION OF NEUROLOGICAL DISORDERS COURSING WITH A COGNITION DEFICIT OR IMPAIRMENT, AND OF NEURODEGENERATIVE DISEASES FUNDACIÓN PARA LA INVESTIGACIÓN MÉDICA APLICADA (ES) 2017-08-17 US claimed
EP-3185903-A1 PRODUCTS FOR THE TREATMENT AND PREVENTION OF NEUROLOGICAL DISORDERS COURSING WITH A COGNITION DEFICIT OR IMPAIRMENT, AND OF NEURODEGENERATIVE DISEASES Fundación para la Investigación Médica Aplicada (ES) 2017-07-05 EP claimed
CN-106604747-A PRODUCTS FOR THE TREATMENT AND PREVENTION OF NEUROLOGICAL DISORDERS COURSING WITH A COGNITION DEFICIT OR IMPAIRMENT, AND OF NEURODEGENERATIVE DISEASES 基础应用医学研究基金会 2017-04-26 CN claimed
EP-2330894-B1 COMPOSITIONS INCLUDING 6-AMINOHEXANOIC ACID DERIVATIVES AS HDAC INHIBITORS REPLIGEN CORP (US) 2016-12-21 EP claimed
US-20160122290-A1 COMPOSITIONS INCLUDING 6-AMINOHEXANOIC ACID DERIVATIVES AS HDAC INHIBITORS REPLIGEN CORPORATION 2016-05-05 US claimed
WO-2016030345-A1 PRODUCTS FOR THE TREATMENT AND PREVENTION OF NEUROLOGICAL DISORDERS COURSING WITH A COGNITION DEFICIT OR IMPAIRMENT, AND OF NEURODEGENERATIVE DISEASES FUNDACIÓN PARA LA INVESTIGACIÓN MÉDICA APLICADA (ES) 2016-03-03 WO claimed
US-9265734-B2 Compositions including 6-aminohexanoic acid derivatives as HDAC inhibitors BIOMARIN PHARMACEUTICAL INC. (US) 2016-02-23 US claimed
US-20120094971-A1 Compositions Including 6-Aminohexanoic Acid Derivatives As HDAC Inhibitors REPLIGEN CORPORATION (US) 2012-04-19 US claimed
EP-2330894-A1 COMPOSITIONS INCLUDING 6-AMINOHEXANOIC ACID DERIVATIVES AS HDAC INHIBITORS REPLIGEN CORPORATION (US) 2011-06-15 EP claimed
WO-2010028192-A1 COMPOSITIONS INCLUDING 6-AMINOHEXANOIC ACID DERIVATIVES AS HDAC INHIBITORS REPLIGEN CORPORATION (US) 2010-03-11 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160122290-A1 COMPOSITIONS INCLUDING 6-AMINOHEXANOIC ACID DERIVATIVES AS HDAC INHIBITORS HDAC1, HDAC5, HDAC2 HDAC3 5/4885HDAC1 1/4885HDAC2 3/4885
US-20170231931-A1 PRODUCTS FOR THE TREATMENT AND PREVENTION OF NEUROLOGICAL DISORDERS COURSING WITH A COGNITION DEFICIT OR IMPAIRMENT, AND OF NEURODEGENERATIVE DISEASES SNCA, PSEN2, PSEN1 HDAC3 3869/4885HDAC1 3531/4885HDAC2 2063/4885
US-20120094971-A1 Compositions Including 6-Aminohexanoic Acid Derivatives As HDAC Inhibitors HDAC1, HDAC5, HDAC2 HDAC3 5/4885HDAC1 1/4885HDAC2 3/4885
US-20260125650-A1 METHODS AND COMPOSITIONS FOR GENERATING HEPATOCYTES WNT3A, GSK3B, GSK3A HDAC3 97/4885HDAC1 71/4885HDAC2 432/4885
US-20250161243-A1 MEF2 TRANSCRIPTIONAL ACTIVATORS TO TREAT NEUROLOGIC CONDITIONS MEF2D, TEAD2, TEAD1 HDAC3 842/4885HDAC1 186/4885HDAC2 117/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.