SCHEMBL529253

SCHEMBL529253

Cc1ccc2ncc(C(=O)O)c(NCCCN(C)C)c2c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.58
KMT2A Q03164 6/20 0.53
MEN1 O00255 4/20 0.53
KDM4E B2RXH2 2/20 0.53
GAA P10253 2/20 0.53
POLB P06746 3/20 0.47
SMN1; SMN2 Q16637 3/20 0.47
RAD52 P43351 3/20 0.46
UHRF1 Q96T88 1/20 0.46
CYP1A2 P05177 1/20 0.46
NPC1 O15118 1/20 0.44
SLC2A1 P11166 1/20 0.44
APOBEC3A P31941 1/20 0.44
RAB9A P51151 1/20 0.44
APOBEC3G Q9HC16 1/20 0.44
TP53 P04637 2/20 0.44
MAPT P10636 2/20 0.44
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43
ATM Q13315 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL530085 0.88 KMT2A (0.50) MAPK1KMT2AMEN1KDM4EGAA
SCHEMBL10282420 0.87 MAPK1 (0.78) MAPK1KMT2AMEN1KDM4EGAA
SCHEMBL529115 0.85 MELK (0.51) MAPK1KMT2AMEN1KDM4EGAA
SCHEMBL530888 0.84 KCNH2 (0.54) MAPK1KMT2AMEN1KDM4EGAA
SCHEMBL531008 0.83 KMT2A (0.46) KMT2AMEN1KDM4EGAAPOLB
SCHEMBL10282210 0.82 MAPT (0.50) KMT2AMEN1KDM4EGAAPOLB
SCHEMBL20435808 0.82 RAD52 (0.50) MAPK1KMT2AMEN1KDM4EGAA
Hydrochloric Acid SCHEMBL529682 0.81 MAPT (0.49) KMT2AMEN1KDM4EGAAPOLB
SCHEMBL530078 0.81 KMT2A (0.44) MAPK1KMT2AMEN1KDM4EGAA
SCHEMBL10282212 0.80 MELK (0.50) MAPK1KMT2AMEN1KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2597955-A1 QUINOLINE DERIVATIVES AND MELK INHIBITORS CONTAINING THE SAME OncoTherapy Science, Inc. (JP) 2013-06-05 EP disclosed
WO-2012016082-A1 QUINOLINE DERIVATIVES AND MELK INHIBITORS CONTAINING THE SAME ONCOTHERAPY SCIENCE, INC. (JP) 2012-02-02 WO disclosed