SCHEMBL5292581

SCHEMBL5292581

C=C(CC)C(=O)O.C=CN1CCCC1=O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.36
KMT2A Q03164 2/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA3 P07451 1/20 0.36
CA4 P22748 1/20 0.36
CA6 P23280 1/20 0.36
CA5A P35218 1/20 0.36
CA7 P43166 1/20 0.36
CA9 Q16790 1/20 0.36
CA13 Q8N1Q1 1/20 0.36
CA14 Q9ULX7 1/20 0.36
CA5B Q9Y2D0 1/20 0.36
INMT O95050 1/20 0.34
TSHR P16473 1/20 0.33
BRD4 O60885 1/20 0.32
BRD2 P25440 1/20 0.32
BLM P54132 1/20 0.31
ALDH1A1 P00352 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Methacrylic Acid SCHEMBL11236958 0.96 LMNA (0.33) LMNAKMT2ACA12CA1CA2
SCHEMBL9551034 0.88 LMNA (0.36) LMNAKMT2ACA12CA1CA2
Propionic Acid SCHEMBL28130435 0.87 LMNA (0.39) LMNAKMT2ACA12CA1CA2
SCHEMBL11857121 0.86 LMNA (0.34) LMNAKMT2ACA12CA1CA2
Itaconate SCHEMBL17687381 0.85 ALOX15 (0.47) LMNAKMT2ATSHRBLMALDH1A1
Methacrylic Acid SCHEMBL9422689 0.84 KMT2A (0.36) LMNAKMT2ACA12CA1CA2
Methacrylic Acid SCHEMBL887731 0.84 KMT2A (0.36) LMNAKMT2ACA12CA1CA2
SCHEMBL5268013 0.84 LMNA (0.35) LMNAKMT2ACA12CA1CA2
SCHEMBL10443872 0.84 LMNA (0.37) LMNAKMT2ATSHRBLMALDH1A1
Methacrylic Acid SCHEMBL6881562 0.83 LMNA (0.33) LMNAKMT2ACA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 22 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1366087-B1 UV-CURABLE, NON-CHLORINATED ADHESION PROMOTERS EASTMAN CHEM CO (US) 2004-08-11 EP claimed
EP-3132084-A2 AQUEOUS SOLUTIONS OF WATER-SOLUBLE POLYMERS AS AN ADJUVANT IN TEXTILE PRE-TREATMENT OF COTTON AND ITS BLENDS WITH SYNTHETIC FIBRES Archroma IP GmbH (CH) 2017-02-22 EP disclosed
WO-2015158437-A2 AQUEOUS SOLUTIONS OF WATER-SOLUBLE POLYMERS AS AN ADJUVANT IN TEXTILE PRE-TREATMENT OF COTTON AND ITS BLENDS WITH SYNTHETIC FIBRES ARCHROMA IP GMBH (CH) 2015-10-22 WO disclosed
US-7199103-B2 Synthetic compounds and compositions with enhanced cell binding THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2007-04-03 US disclosed
WO-2007002469-A2 THERAPEUTIC COMPOSITIONS AND METHODS USING TRANSFORMING GROWTH FACTOR-BETA MIMICS BHATNAGAR RAJENDRA S (US) 2007-01-04 WO disclosed
US-20060293228-A1 Therapeutic compositions and methods using transforming growth factor-beta mimics BHATNAGAR RAJENDRA S 2006-12-28 US disclosed
EP-0951472-B1 PEPTIDE COMPOSITIONS WITH GROWTH FACTOR-LIKE ACTIVITY UNIV CALIFORNIA (US) 2006-08-09 EP disclosed
US-20050164944-A1 Synthetic compounds and compositions with enhanced cell binding THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2005-07-28 US disclosed
US-6818620-B2 POLYPEPTIDES THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2004-11-16 US disclosed
US-20020037853-A1 Synthetic compounds and compositions with enhanced cell binding THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2002-03-28 US disclosed
EP-0824545-B1 PEPTIDE COMPOSITIONS WITH GROWTH FACTOR-LIKE ACTIVITY UNIV CALIFORNIA (US) 1999-12-08 EP disclosed
US-5958428-A SYNTHETIC PEPTIDES THAT MIMIC THE CONFORMATION NECESSARY FOR RECOGNITION AND DOCKING OF COLLAGEN BINDING SPECIES (SUCH AS CELL SURFACE RECEPTORS FOR COLLAGEN AND FIBRONECTIN) AND HAVE THE AMINO ACID RESIDUES-ILE-ALA-FOLDED IN A .BETA.-BEND THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1999-09-28 US disclosed
US-5780436-A WOUND HEALING HEXA- AND HEPTAPEPTIDES THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1998-07-14 US disclosed
US-5674848-A PACKING MATERIAL THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1997-10-07 US disclosed
US-5661127-A HEPTAPEPTIDE FOR USE WITH BIOCOMPATIBLE MATRICES IN TISSUE REPAIR OR IMPLANTS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1997-08-26 US disclosed
US-5635482-A IMPLANT COMPRISING MATRIX FORMED OF BIOMATERIAL AND PEPTIDE HAVING ENHANCED CELL BINDING WITH RESPECT TO COLLAGEN THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1997-06-03 US disclosed
EP-0618802-A4 SYNTHETIC COMPOUNDS AND COMPOSITIONS WITH ENHANCED CELL BINDING. UNIV CALIFORNIA (US) 1996-12-18 EP disclosed
EP-0618802-A1 SYNTHETIC COMPOUNDS AND COMPOSITIONS WITH ENHANCED CELL BINDING THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1994-10-12 EP disclosed
US-5354736-A Peridontal repair mixture composed of hydroxyapatite particles coated with synthetic peptides REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1994-10-11 US disclosed
WO-1993011781-A1 SYNTHETIC COMPOUNDS AND COMPOSITIONS WITH ENHANCED CELL BINDING THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1993-06-24 WO disclosed