SCHEMBL5293012

SCHEMBL5293012

CC1CCCCC(N2N=C(C3CCCCC3)c3ccccc3NC2=O)CC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.37
ALDH1A1 P00352 6/20 0.34
HPGD P15428 5/20 0.34
KDM4E B2RXH2 4/20 0.34
SMN1; SMN2 Q16637 3/20 0.34
RAB9A P51151 2/20 0.34
NPSR1 Q6W5P4 1/20 0.34
HSD17B10 Q99714 2/20 0.33
MEN1 O00255 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
STAT3 P40763 1/20 0.33
KMT2A Q03164 1/20 0.33
GAA P10253 1/20 0.33
CNR1 P21554 1/20 0.32
OPRM1 P35372 2/20 0.32
OPRD1 P41143 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5324581 0.92 CES2 (0.41) CES2ALDH1A1HPGDKDM4ESMN1; SMN2
SCHEMBL5320501 0.92 CES2 (0.41) CES2ALDH1A1HPGDKDM4ESMN1; SMN2
SCHEMBL5324527 0.92 CES2 (0.41) CES2ALDH1A1HPGDKDM4ESMN1; SMN2
SCHEMBL5325094 0.92 CES2 (0.41) CES2ALDH1A1HPGDKDM4ESMN1; SMN2
SCHEMBL5321802 0.92 CES2 (0.41) CES2ALDH1A1HPGDKDM4ESMN1; SMN2
SCHEMBL5328233 0.85 OPRM1 (0.35) CES2ALDH1A1HPGDKDM4ENPSR1
SCHEMBL5328236 0.85 OPRM1 (0.35) CES2ALDH1A1HPGDKDM4ENPSR1
SCHEMBL5321151 0.85 CYP2D6 (0.39) CES2ALDH1A1HPGDKDM4ESMN1; SMN2
SCHEMBL5321156 0.85 CYP2D6 (0.39) CES2ALDH1A1HPGDKDM4ESMN1; SMN2
SCHEMBL5322846 0.84 PTH1R (0.38) CES2ALDH1A1HPGDKDM4ENPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006129120-A9 BENZOTRIAZEPINONE DERIVATIVES JAMES BLACK FOUNDATION (GB) 2007-03-22 WO disclosed
WO-2006129120-A2 BENZOTRIAZEPINONE DERIVATIVES JAMES BLACK FOUNDATION (GB) 2006-12-07 WO disclosed