SCHEMBL529904

SCHEMBL529904

NCC(=O)c1cnc2ccccc2c1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MGAM O43451 1/20 0.65
CFTR P13569 1/20 0.58
RAB9A P51151 4/20 0.49
TOP2A P11388 2/20 0.48
TOP2B Q02880 2/20 0.48
BCAT1 P54687 1/20 0.48
KDM4E B2RXH2 2/20 0.48
KMT2A Q03164 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
KDR P35968 1/20 0.48
MAP4K4 O95819 1/20 0.46
CSNK1G2 P78368 1/20 0.46
CLK4 Q9HAZ1 1/20 0.46
MKNK2 Q9HBH9 1/20 0.46
MAP4K5 Q9Y4K4 1/20 0.46
NPC1 O15118 2/20 0.44
ALDH1A1 P00352 1/20 0.44
CYP1A2 P05177 1/20 0.44
DPP4 P27487 1/20 0.44
HPGDS O60760 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7100632 0.84 MGAM (0.61) MGAMCFTRRAB9ATOP2ATOP2B
SCHEMBL9700485 0.84 MGAM (0.61) MGAMCFTRRAB9ATOP2ATOP2B
SCHEMBL21296699 0.83 MGAM (0.65) MGAMCFTRRAB9ATOP2ATOP2B
SCHEMBL8270577 0.83 MGAM (0.65) MGAMCFTRRAB9ATOP2ATOP2B
SCHEMBL4817449 0.83 MGAM (0.65) MGAMCFTRRAB9ATOP2ATOP2B
SCHEMBL5363975 0.82 MGAM (0.68) MGAMCFTRRAB9ATOP2ATOP2B
SCHEMBL29362497 0.81 MGAM (0.71) MGAMCFTRRAB9ATOP2ATOP2B
SCHEMBL23372 0.81 MGAM (0.71) MGAMCFTRRAB9ATOP2ATOP2B
SCHEMBL12505008 0.81 CFTR (0.68) MGAMCFTRRAB9ATOP2ATOP2B
SCHEMBL9361658 0.81 MGAM (0.61) MGAMCFTRRAB9ATOP2ATOP2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2597955-A1 QUINOLINE DERIVATIVES AND MELK INHIBITORS CONTAINING THE SAME OncoTherapy Science, Inc. (JP) 2013-06-05 EP disclosed
EP-2471786-A1 AMINOPYRAZOLE DERIVATIVE Chugai Seiyaku Kabushiki Kaisha (JP) 2012-07-04 EP disclosed
WO-2012016082-A1 QUINOLINE DERIVATIVES AND MELK INHIBITORS CONTAINING THE SAME ONCOTHERAPY SCIENCE, INC. (JP) 2012-02-02 WO disclosed
WO-2011016528-A1 AMINOPYRAZOLE DERIVATIVE 中外製薬株式会社 (JP) 2011-02-10 WO disclosed