SCHEMBL529996

SCHEMBL529996

CC(C)(C)OC(=O)N(c1ncc(N)cn1)C1CCNC1

nearest known ligand 0.36

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 20/20 0.36
SLC6A2 P23975 19/20 0.36
SLC6A3 Q01959 15/20 0.36
CYP2D6 P10635 5/20 0.34
KCNH2 Q12809 4/20 0.34
CHRM3 P20309 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28329578 0.85 SLC6A4 (0.39) SLC6A4SLC6A2SLC6A3CYP2D6KCNH2
SCHEMBL3635111 0.81 SLC6A4 (0.35) SLC6A4SLC6A2SLC6A3CYP2D6KCNH2
SCHEMBL3635108 0.81 SLC6A4 (0.35) SLC6A4SLC6A2SLC6A3CYP2D6KCNH2
SCHEMBL29017156 0.80 GPR119 (0.38) SLC6A4SLC6A2SLC6A3CYP2D6
SCHEMBL18142028 0.79 SLC6A4 (0.35) SLC6A4SLC6A2SLC6A3CYP2D6KCNH2
SCHEMBL529417 0.79 RPLP1 (0.36) KCNH2
SCHEMBL529544 0.79 RPLP1 (0.36) KCNH2
SCHEMBL2597129 0.79 EP300 (0.34) SLC6A4SLC6A2SLC6A3CYP2D6KCNH2
SCHEMBL26697116 0.78 SLC6A4 (0.34) SLC6A4SLC6A2SLC6A3CYP2D6KCNH2
SCHEMBL4439873 0.77 SLC6A4 (0.36) SLC6A4SLC6A2SLC6A3CYP2D6KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2597955-A1 QUINOLINE DERIVATIVES AND MELK INHIBITORS CONTAINING THE SAME OncoTherapy Science, Inc. (JP) 2013-06-05 EP disclosed
WO-2012016082-A1 QUINOLINE DERIVATIVES AND MELK INHIBITORS CONTAINING THE SAME ONCOTHERAPY SCIENCE, INC. (JP) 2012-02-02 WO disclosed