SCHEMBL5300761

SCHEMBL5300761

Cc1ccc(C)c(C(C)(C)N)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.46
TDP1 Q9NUW8 3/20 0.46
TAAR1 Q96RJ0 1/20 0.39
SMN1; SMN2 Q16637 3/20 0.38
HSD17B10 Q99714 3/20 0.38
KDM4E B2RXH2 2/20 0.38
GAA P10253 2/20 0.38
LMNA P02545 1/20 0.38
HPGD P15428 1/20 0.38
TP53 P04637 2/20 0.37
ALOX15 P16050 2/20 0.37
CYP3A4 P08684 1/20 0.37
THRB P10828 1/20 0.37
CYP1A2 P05177 2/20 0.36
CYP2A6 P11509 2/20 0.36
POLB P06746 2/20 0.34
CA2 P00918 1/20 0.34
TYR P14679 1/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23211226 0.86 ALDH1A1 (0.46) ALDH1A1TDP1TAAR1SMN1; SMN2HSD17B10
SCHEMBL17972841 0.81 CASR (0.41) ALDH1A1TDP1TAAR1SMN1; SMN2HSD17B10
SCHEMBL15200202 0.80 ALDH1A1 (0.41) ALDH1A1TDP1TAAR1SMN1; SMN2HSD17B10
SCHEMBL16105750 0.80 TDP1 (0.44) ALDH1A1TDP1TAAR1SMN1; SMN2HSD17B10
SCHEMBL3166363 0.80 ALDH1A1 (0.48) ALDH1A1TDP1TAAR1SMN1; SMN2HSD17B10
SCHEMBL18536951 0.79 SMN1; SMN2 (0.46) ALDH1A1TDP1TAAR1SMN1; SMN2HSD17B10
SCHEMBL16579354 0.77 SMN1; SMN2 (0.36) ALDH1A1TDP1SMN1; SMN2LMNAHPGD
SCHEMBL29939083 0.77 SMN1; SMN2 (0.40) ALDH1A1TDP1TAAR1SMN1; SMN2HSD17B10
SCHEMBL16579355 0.77 CYP3A4 (0.50) ALDH1A1TDP1SMN1; SMN2KDM4EGAA
SCHEMBL10328480 0.76 SMN1; SMN2 (0.42) ALDH1A1TDP1TAAR1SMN1; SMN2HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007016190-A2 ANTIPARKINSONIAN ACTION OF PHENYLISOPROPYLAMINES DUKE UNIVERSITY (US) 2007-02-08 WO claimed
US-20070027208-A1 Antiparkinsonian Action of Phenylisopropylamines NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2007-02-01 US claimed
US-20160221948-A1 NITROGEN-CONTAINING SATURATED HETEROCYCLIC COMPOUND SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2016-08-04 US disclosed
US-20160221948-A1 NITROGEN-CONTAINING SATURATED HETEROCYCLIC COMPOUND SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2016-08-04 US disclosed
US-20150025063-A1 Antiparkinsonian Action of Phenylisopropylamines UNIV DUKE (US) 2015-01-22 US disclosed
US-8877802-B2 Antiparkinsonian action of phenylisopropylamines Duke Univerity (US) 2014-11-04 US disclosed
WO-2007016190-A2 ANTIPARKINSONIAN ACTION OF PHENYLISOPROPYLAMINES DUKE UNIVERSITY (US) 2007-02-08 WO disclosed
US-20070027208-A1 Antiparkinsonian Action of Phenylisopropylamines NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2007-02-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160221948-A1 NITROGEN-CONTAINING SATURATED HETEROCYCLIC COMPOUND H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16, H1-4, HRH4 ALDH1A1 2734/4885TDP1 4532/4885TAAR1 1517/4885
US-20070027208-A1 Antiparkinsonian Action of Phenylisopropylamines PNMT, SNCA, COMT ALDH1A1 926/4885TDP1 716/4885TAAR1 1075/4885
US-20150025063-A1 Antiparkinsonian Action of Phenylisopropylamines PNMT, SNCA, COMT ALDH1A1 926/4885TDP1 716/4885TAAR1 1075/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.