SCHEMBL5300822

SCHEMBL5300822

CC(Cc1ccccc1)(NC(=O)CN)c1ccc(O)cc1

nearest known ligand 0.84

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.84
CYP1A2 P05177 1/20 0.84
RECQL P46063 1/20 0.84
MAPK1 P28482 1/20 0.82
BLM P54132 1/20 0.44
KIF11 P52732 2/20 0.44
ESR1 P03372 4/20 0.41
ESR2 Q92731 4/20 0.41
ALDH1A1 P00352 3/20 0.41
CYP2C19 P33261 2/20 0.40
CYP2C9 P11712 1/20 0.40
OPRM1 P35372 1/20 0.40
OPRD1 P41143 1/20 0.40
OPRK1 P41145 1/20 0.40
POLB P06746 1/20 0.40
GAA P10253 1/20 0.40
LTA4H P09960 1/20 0.39
MEN1 O00255 1/20 0.39
TSHR P16473 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5300046 0.94 CYP3A4 (0.84) CYP3A4CYP1A2RECQLMAPK1BLM
Fumaric Acid SCHEMBL8866741 0.94 CYP3A4 (0.74) CYP3A4CYP1A2RECQLMAPK1BLM
Maleic Acid SCHEMBL8866733 0.94 CYP3A4 (0.74) CYP3A4CYP1A2RECQLMAPK1BLM
SCHEMBL5306503 0.93 CYP3A4 (0.71) CYP3A4CYP1A2RECQLMAPK1BLM
Acetic Acid SCHEMBL8866866 0.92 CYP3A4 (0.70) CYP3A4CYP1A2RECQLMAPK1BLM
Remacemide SCHEMBL151148 0.91 CYP1A2 (1.00) CYP3A4CYP1A2RECQLMAPK1ALDH1A1
Remacemide SCHEMBL20769836 0.91 CYP1A2 (1.00) CYP3A4CYP1A2RECQLMAPK1ALDH1A1
Remacemide SCHEMBL635940 0.90 MAPK1 (1.00) CYP3A4CYP1A2RECQLMAPK1ALDH1A1
SCHEMBL9054250 0.89 CYP3A4 (0.84) CYP3A4CYP1A2RECQLMAPK1KIF11
Fumaric Acid SCHEMBL8866366 0.89 CYP3A4 (0.74) CYP3A4CYP1A2RECQLMAPK1BLM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007017652-A2 ARYLAKYLAMINES FOR THE TREATMENT OF CANCER ASTRAZENECA AB (SE) 2007-02-15 WO claimed
EP-0356035-B1 Arylkalkyl-amines and -amides having anticonvulsant and neuroprotective properties ASTRA AB (SE) 1996-03-13 EP claimed
WO-1991011995-A1 ARYLALKYL-AMINES AND -AMIDES HAVING ANTICONVULSANT AND NEUROPROTECTIVE PROPERTIES FISONS CORPORATION (US) 1991-08-22 WO claimed
EP-0356035-A2 Arylkalkyl-amines and -amides having anticonvulsant and neuroprotective properties Astra Aktiebolag (SE) 1990-02-28 EP claimed
WO-2007017652-A2 ARYLAKYLAMINES FOR THE TREATMENT OF CANCER ASTRAZENECA AB (SE) 2007-02-15 WO disclosed