SCHEMBL530104

SCHEMBL530104

CC(C)(C)OC(=O)c1ccc(C(=O)NNc2ncccc2Br)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.52
ALDH1A1 P00352 3/20 0.46
POLB P06746 1/20 0.46
TLR7 Q9NYK1 7/20 0.41
RAB9A P51151 4/20 0.39
NPC1 O15118 3/20 0.39
HPGD P15428 2/20 0.39
PKM P14618 1/20 0.39
CDK5 Q00535 1/20 0.39
PAX8 Q06710 1/20 0.39
CDK5R1 Q15078 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39
CA14 Q9ULX7 1/20 0.39
STAT3 P40763 1/20 0.38
ABCG2 Q9UNQ0 1/20 0.38
NAMPT P43490 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12887986 0.86 NAMPT (0.56) GAAALDH1A1POLBNAMPT
SCHEMBL1179500 0.76 GAA (0.45) GAAALDH1A1POLBTLR7RAB9A
SCHEMBL16600343 0.76 STAT3 (0.51) RAB9ANPC1SMN1; SMN2STAT3NAMPT
SCHEMBL29476654 0.73 METAP1 (0.46) RAB9ANPC1SMN1; SMN2NAMPT
SCHEMBL623831 0.73 METAP1 (0.46) RAB9ANPC1SMN1; SMN2NAMPT
SCHEMBL1155947 0.72 LMNA (0.46) GAAALDH1A1POLBTLR7RAB9A
SCHEMBL21358025 0.71 GABRA1 (0.42) ALDH1A1POLBRAB9ANPC1
SCHEMBL24602868 0.70 HDAC1 (0.60) CA12CA1CA2CA9CA14
SCHEMBL456000 0.69 MEN1 (0.44) GAAALDH1A1POLBRAB9ANPC1
SCHEMBL16879880 0.69 GAA (0.47) GAAALDH1A1POLBRAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012015693-A1 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2012-02-02 WO disclosed