SCHEMBL5301510

SCHEMBL5301510

NC(=O)c1cc(Oc2ccc(C(=O)Nc3c(-c4ccc(F)cc4)cc[nH]c3=O)cc2F)ccn1

nearest known ligand 0.44

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MET P08581 16/20 0.44
KDR P35968 6/20 0.42
BCL9 O00512 1/20 0.41
CTNNB1 P35222 1/20 0.41
BRD4 O60885 1/20 0.40
AXL P30530 1/20 0.40
HIPK4 Q8NE63 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5306561 0.81 MET (0.43) METKDRAXLHIPK4
SCHEMBL1269377 0.74 MET (0.58) METKDRAXL
SCHEMBL1269426 0.72 MET (0.49) METKDRAXL
SCHEMBL5157575 0.69 AXL (0.44) METKDRAXLHIPK4
SCHEMBL3552329 0.69 MET (0.69) METKDRAXL
SCHEMBL1137174 0.68 MET (0.48) METKDRAXL
SCHEMBL1137376 0.68 KDR (0.64) METKDRAXLHIPK4
SCHEMBL29757310 0.68 GCK (0.56) METKDRAXL
SCHEMBL23913769 0.66 P2RX3 (0.53)
SCHEMBL29757282 0.66 P2RX3 (0.53)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007035428-A1 MET KINASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2007-03-29 WO disclosed