SCHEMBL5302192

SCHEMBL5302192

CS(=O)(=O)c1ccc(-c2ccc(N)c(C#N)c2)cc1

nearest known ligand 0.49

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 9/20 0.49
IKBKB O14920 1/20 0.46
CHUK O15111 1/20 0.46
DHFR P00374 1/20 0.44
PTGS2 P35354 2/20 0.44
G6PD P11413 1/20 0.44
IDE P14735 1/20 0.44
KIF11 P52732 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2577731 0.86 G6PD (0.53) LRRK2IKBKBCHUKPTGS2G6PD
SCHEMBL903994 0.81 LRRK2 (0.49) LRRK2PTGS2KIF11
SCHEMBL5072719 0.80 TDP1 (0.48)
SCHEMBL17674151 0.80 LRRK2 (0.46) LRRK2IKBKBCHUKPTGS2KIF11
SCHEMBL8320176 0.79 MEN1 (0.56) LRRK2DHFRPTGS2G6PDIDE
SCHEMBL3583094 0.78 AR (0.53)
SCHEMBL31037588 0.77 CYP3A4 (0.46) KIF11
SCHEMBL14496780 0.76 G6PD (0.49) LRRK2IKBKBCHUKPTGS2G6PD
SCHEMBL5302056 0.75 MCL1 (0.50) IKBKB
SCHEMBL14191689 0.74 TSHR (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007025575-A1 O-HYDROXY- AND O-AMINO BENZAMIDE DERIVATIVES AS IKK2 INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2007-03-08 WO disclosed