SCHEMBL5306352

SCHEMBL5306352

O=C(O)COCC(=O)Nc1ccn[nH]1

nearest known ligand 0.55

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.55
ALDH1A1 P00352 1/20 0.42
TSHR P16473 1/20 0.42
CYP4F2 P78329 1/20 0.40
CYP4A11 Q02928 1/20 0.40
KMT2A Q03164 1/20 0.39
FFAR2 O15552 1/20 0.39
CHRNB2 P17787 1/20 0.39
CHRNA4 P43681 1/20 0.39
EGFR P00533 1/20 0.38
ALPL P05186 1/20 0.38
KDM4E B2RXH2 1/20 0.38
HCAR2 Q8TDS4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7854147 0.86 PKM (0.57) PKMKMT2AFFAR2CHRNB2CHRNA4
SCHEMBL12974928 0.82 PKM (0.53) PKMFFAR2CHRNB2CHRNA4EGFR
SCHEMBL2661353 0.75 PKM (0.67) PKMALDH1A1KMT2AFFAR2CHRNB2
SCHEMBL4383929 0.75 PKM (0.58) PKMFFAR2CHRNB2CHRNA4EGFR
SCHEMBL1012929 0.74
SCHEMBL4561823 0.72 PKM (0.63) PKMFFAR2EGFR
SCHEMBL2402889 0.69 PKM (0.44) PKMFFAR2EGFRHCAR2
SCHEMBL19905402 0.69 ALDH1A1 (0.59) ALDH1A1KMT2AKDM4E
SCHEMBL3994333 0.69
SCHEMBL3451050 0.69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1855672-A1 HIV PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2007-11-21 EP disclosed
WO-2006104646-A1 HIV PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2006-10-05 WO disclosed