SCHEMBL530637

SCHEMBL530637

CCOC(=O)c1ccc(-n2c(=O)[nH]c3cccnc32)cc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.65
GAA P10253 2/20 0.65
NPC1 O15118 2/20 0.65
HPGD P15428 3/20 0.51
HTT P42858 2/20 0.51
MAT2A P31153 1/20 0.48
MAPT P10636 3/20 0.47
ALDH1A1 P00352 2/20 0.47
HSD17B10 Q99714 2/20 0.47
ALOX15 P16050 1/20 0.47
HSP90AA1 P07900 1/20 0.46
CACNA1B Q00975 1/20 0.46
APBA1 Q02410 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
DAO P14920 1/20 0.46
ELANE P08246 1/20 0.46
LMNA P02545 1/20 0.45
KDM4E B2RXH2 1/20 0.44
POLB P06746 3/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30615622 0.84 DAO (0.54) SMN1; SMN2GAANPC1MAPTALDH1A1
SCHEMBL21464285 0.82 CYP2D6 (0.48) SMN1; SMN2NPC1HTTMAPTALDH1A1
SCHEMBL527382 0.81 SMN1; SMN2 (0.56) SMN1; SMN2GAANPC1HPGDHTT
SCHEMBL527340 0.81 DAO (0.54) SMN1; SMN2HPGDMAPTALDH1A1NPSR1
SCHEMBL1699095 0.81 DAO (0.62) HPGDMAPTALDH1A1DAO
SCHEMBL2256170 0.81 SMN1; SMN2 (0.78) SMN1; SMN2GAANPC1HPGDHTT
SCHEMBL11554147 0.80 ALDH1A1 (0.58) HPGDALDH1A1DAOLMNAKDM4E
SCHEMBL30615419 0.80 NPC1 (0.42) SMN1; SMN2GAANPC1MAT2AMAPT
SCHEMBL28487985 0.80 NPC1 (0.42) SMN1; SMN2GAANPC1MAT2AMAPT
SCHEMBL1699133 0.77 DAO (0.58) ALDH1A1HSP90AA1DAO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012015693-A1 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2012-02-02 WO disclosed