SCHEMBL530809

SCHEMBL530809

CC(N)C(=O)c1cnc2ccccc2c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MGAM O43451 1/20 0.61
CFTR P13569 1/20 0.49
MAP4K4 O95819 1/20 0.47
CSNK1G2 P78368 1/20 0.47
CLK4 Q9HAZ1 1/20 0.47
MKNK2 Q9HBH9 1/20 0.47
MAP4K5 Q9Y4K4 1/20 0.47
CYP1A2 P05177 2/20 0.46
BCAT1 P54687 1/20 0.46
TOP2A P11388 1/20 0.46
TOP2B Q02880 1/20 0.46
KDR P35968 1/20 0.46
DPP4 P27487 1/20 0.45
HPGDS O60760 1/20 0.45
KDM4E B2RXH2 2/20 0.45
RAB9A P51151 2/20 0.45
NPC1 O15118 1/20 0.45
MITF O75030 1/20 0.45
XBP1 P17861 1/20 0.45
PAX8 Q06710 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2625196 0.87 MGAM (0.65) MGAMCFTRMAP4K4CSNK1G2CLK4
SCHEMBL27784603 0.82 MGAM (0.67) MGAMCFTRMAP4K4CSNK1G2CLK4
SCHEMBL10350097 0.80 MGAM (0.59) MGAMCFTRMAP4K4CSNK1G2CLK4
SCHEMBL23372 0.78 MGAM (0.71) MGAMCFTRMAP4K4CSNK1G2CLK4
SCHEMBL530761 0.78 MGAM (0.71) MGAMCFTRMAP4K4CSNK1G2CLK4
SCHEMBL29684771 0.78 MGAM (0.71) MGAMCFTRMAP4K4CSNK1G2CLK4
SCHEMBL29362497 0.78 MGAM (0.71) MGAMCFTRMAP4K4CSNK1G2CLK4
SCHEMBL7371232 0.78 MGAM (0.76) MGAMCFTRMAP4K4CSNK1G2CLK4
SCHEMBL15309423 0.78 MGAM (0.56) MGAMCFTRMAP4K4CSNK1G2CLK4
SCHEMBL12043740 0.77 HPGDS (0.67) MGAMCYP1A2BCAT1KDRHPGDS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2597955-A1 QUINOLINE DERIVATIVES AND MELK INHIBITORS CONTAINING THE SAME OncoTherapy Science, Inc. (JP) 2013-06-05 EP disclosed
WO-2012016082-A1 QUINOLINE DERIVATIVES AND MELK INHIBITORS CONTAINING THE SAME ONCOTHERAPY SCIENCE, INC. (JP) 2012-02-02 WO disclosed